SCHEMBL5226889

SCHEMBL5226889

CC(C)(O)c1cccc2nc(-c3ccc(O)cc3)oc12

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CEPT1 Q9Y6K0 1/20 0.53
ESR2 Q92731 18/20 0.50
ESR1 P03372 15/20 0.50
HDAC6 Q9UBN7 1/20 0.47
DHODH Q02127 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21776932 0.87 CEPT1 (0.52) CEPT1ESR2ESR1DHODH
SCHEMBL3919291 0.85 CEPT1 (0.50) CEPT1HDAC6DHODH
SCHEMBL2402116 0.83 ESR2 (0.64) ESR2ESR1HDAC6
SCHEMBL14266178 0.79 ESR2 (0.52) ESR2ESR1HDAC6DHODH
SCHEMBL29819729 0.76 DHODH (0.54) CEPT1ESR2ESR1DHODH
SCHEMBL29819687 0.76 DHODH (0.54) CEPT1ESR2ESR1DHODH
SCHEMBL21776901 0.73 CEPT1 (0.56) CEPT1
SCHEMBL21237208 0.73 ALDH1A1 (0.56) CEPT1DHODH
SCHEMBL28616475 0.73 ESR2 (0.56) ESR2ESR1HDAC6
SCHEMBL10236256 0.72 NPC1 (0.48) ESR2ESR1HDAC6DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017031276-A1 METHODS OF PROVIDING NEUROPROTECTIVE THERAPY RELATED TO ADMINISTERING AN ESTROGEN RECEPTOR BETA LIGAND THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2017-02-23 WO disclosed
EP-1781628-A2 PRODRUG SUBSTITUTED BENZOXAZOLES AS ESTROGENIC AGENTS Wyeth a Corporation of the State of Delaware (US) 2007-05-09 EP disclosed
WO-2006026316-A2 PRODRUG SUBSTITUTED BENZOXAZOLES AS ESTROGENIC AGENTS WYETH (US) 2006-03-09 WO disclosed