SCHEMBL5227313

SCHEMBL5227313

C[C@H](N)C(=O)N[C@@H]1C(=O)Nc2cc(F)ccc2C[C@@H]1c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.36
SOAT1 P35610 1/20 0.36
SMYD3 Q9H7B4 1/20 0.36
MAPK1 P28482 1/20 0.35
RECQL P46063 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
GRM7 Q14831 1/20 0.35
HSD17B2 P37059 2/20 0.35
PAX8 Q06710 1/20 0.34
RIPK1 Q13546 1/20 0.34
XIAP P98170 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
AKR1B1 P15121 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5227301 0.84 KDM1A (0.46) ALDH1A1HSD17B2RIPK1MEN1KMT2A
SCHEMBL3345083 0.82 PSEN1 (0.49)
SCHEMBL3346480 0.81 PSEN1 (0.38) SOAT1HSD17B2XIAP
SCHEMBL3346473 0.81 PSEN1 (0.38) SOAT1HSD17B2XIAP
SCHEMBL3343323 0.81 SOAT1 (0.35) ALDH1A1SOAT1HSD17B2MEN1KMT2A
SCHEMBL3343463 0.77 ALDH1A1 (0.40) ALDH1A1MAPK1HSD17B2MEN1KMT2A
SCHEMBL14260860 0.77 ALDH1A1 (0.53) ALDH1A1RECQLMEN1KMT2A
SCHEMBL4117171 0.76 TP53 (0.39) ALDH1A1MAPK1HSD17B2GAA
SCHEMBL8338572 0.76 KDM4E (0.40) ALDH1A1MAPK1RECQLHSD17B2AKR1B1
SCHEMBL14260858 0.76 KDM4E (0.40) ALDH1A1MAPK1RECQLHSD17B2AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1845089-A1 Novel lactams and uses thereof AstraZeneca AB (SE) 2007-10-17 EP disclosed