SCHEMBL5229878

SCHEMBL5229878

CC(C)(C)OC(=O)Nc1ccc2sc(COC(=O)OCc3nc4c(F)c(NC(=O)OC(C)(C)C)ccc4s3)nc2c1F

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.35
METAP1 P53582 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34
KCNQ4 P56696 3/20 0.34
KCNQ5 Q9NR82 3/20 0.34
TRPV1 Q8NER1 1/20 0.34
LCK P06239 6/20 0.33
SYK P43405 1/20 0.33
BRAF P15056 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
LMNA P02545 1/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5229881 0.93 CYP17A1 (0.35) CYP17A1METAP1CYP1A2CYP2C19KCNQ4
SCHEMBL18180255 0.82 NPC1 (0.39) CYP17A1METAP1LCKBRAFLMNA
SCHEMBL5226064 0.76 TRPV1 (0.55) CYP1A2CYP2C19TRPV1
SCHEMBL5122450 0.74 CYP17A1 (0.32) CYP17A1METAP1KCNQ4KCNQ5BRAF
SCHEMBL5226068 0.68 TRPV1 (0.52) CYP1A2CYP2C19TRPV1
SCHEMBL29069807 0.67 CYP17A1 (0.41) CYP17A1METAP1KCNQ4KCNQ5RXFP1
SCHEMBL10187654 0.66 CYP17A1 (0.43) CYP17A1METAP1KCNQ4KCNQ5LCK
SCHEMBL28707071 0.66 CYP17A1 (0.43) CYP17A1METAP1KCNQ4KCNQ5RXFP1
SCHEMBL30126587 0.66 CYP17A1 (0.39) CYP17A1METAP1CYP2C19KCNQ4KCNQ5
SCHEMBL30466622 0.66 GAA (0.46) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1799661-A1 NEW HYDROXYMETHYLBENZOTHIAZOLES AMIDES AstraZeneca AB (SE) 2007-06-27 EP disclosed
WO-2006038871-A1 NEW HYDROXYMETHYLBENZOTHIAZOLES AMIDES ASTRAZENECA AB (SE) 2006-04-13 WO disclosed