SCHEMBL5229972

SCHEMBL5229972

Cc1ccc(Nc2ccccc2NC(=O)c2ccc(C(C)(C)C)cc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.59
RAB9A P51151 7/20 0.59
ALDH1A1 P00352 1/20 0.59
GLA P06280 1/20 0.59
ATM Q13315 1/20 0.59
L3MBTL1 Q9Y468 1/20 0.59
MAPT P10636 3/20 0.56
RECQL P46063 1/20 0.56
CA1 P00915 1/20 0.56
CA2 P00918 1/20 0.56
NR1H4 Q96RI1 4/20 0.54
PPARG P37231 3/20 0.54
PPARA Q07869 1/20 0.54
SMN1; SMN2 Q16637 3/20 0.53
HDAC3 O15379 1/20 0.52
HDAC11 Q96DB2 1/20 0.52
HDAC8 Q9BY41 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
KCNK9 Q9NPC2 1/20 0.52
TRPV1 Q8NER1 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5223950 0.84 NR1H4 (0.71) NPC1RAB9ANR1H4PPARGPPARA
SCHEMBL1687867 0.82 NPC1 (0.79) NPC1RAB9AMAPTCA1CA2
SCHEMBL5223315 0.82 RAB9A (0.73) NPC1RAB9AALDH1A1GLAATM
SCHEMBL7291713 0.82 NPC1 (0.79) NPC1RAB9AMAPTCA1CA2
SCHEMBL7293746 0.82 NPC1 (0.79) NPC1RAB9AMAPTCA1CA2
SCHEMBL12636930 0.80 NPC1 (0.61) NPC1RAB9AALDH1A1MAPTSMN1; SMN2
SCHEMBL13744870 0.80 CA2 (0.58) NPC1RAB9AMAPTRECQLCA1
SCHEMBL7295495 0.79 POLB (0.72) NPC1RAB9AALDH1A1GLAATM
SCHEMBL28199719 0.79 KCNK9 (0.58) NPC1RAB9AALDH1A1GLAATM
SCHEMBL17546531 0.78 AKR1C3 (0.45) NPC1RAB9AALDH1A1GLAATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1014962-A4 ANTITHROMBOTIC AGENTS LILLY CO ELI (US) 2007-06-27 EP disclosed
EP-1014962-A1 ANTITHROMBOTIC AGENTS ELI LILLY AND COMPANY (US) 2000-07-05 EP disclosed
WO-1999000121-A1 ANTITHROMBOTIC AGENTS ELI LILLY AND COMPANY (US) 1999-01-07 WO disclosed