SCHEMBL5230093

SCHEMBL5230093

O=C(NCCCc1cccc(N2CC3CN(C(=O)c4c(F)cccc4Cl)CC3C2)c1)c1cc(F)cc(F)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 5/20 0.39
HCRTR2 O43614 5/20 0.39
SIGMAR1 Q99720 1/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
LIPG Q9Y5X9 1/20 0.37
POLB P06746 1/20 0.37
NAMPT P43490 2/20 0.37
MAPK8 P45983 1/20 0.36
MAPK10 P53779 1/20 0.36
CHRM1 P11229 1/20 0.36
RORC P51449 1/20 0.36
LMNA P02545 2/20 0.36
TP53 P04637 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5230652 0.94 NAMPT (0.42) HCRTR1HCRTR2SIGMAR1NPC1RAB9A
SCHEMBL5240254 0.94 NPC1 (0.46) HCRTR1HCRTR2SIGMAR1NPC1RAB9A
SCHEMBL5239318 0.93 NPC1 (0.43) HCRTR1HCRTR2SIGMAR1NPC1RAB9A
SCHEMBL5233648 0.93 HCRTR1 (0.42) HCRTR1HCRTR2SIGMAR1NPC1RAB9A
SCHEMBL5231455 0.92 NAMPT (0.40) HCRTR1HCRTR2SIGMAR1NPC1RAB9A
SCHEMBL5237555 0.92 NAMPT (0.40) HCRTR1HCRTR2SIGMAR1NPC1RAB9A
SCHEMBL5235222 0.92 HTR1A (0.41) HCRTR1HCRTR2SIGMAR1NPC1RAB9A
SCHEMBL5239914 0.91 HCRTR1 (0.42) HCRTR1HCRTR2SIGMAR1NPC1RAB9A
SCHEMBL5233573 0.90 HSD17B10 (0.41) HCRTR1HCRTR2NPC1RAB9APOLB
SCHEMBL5236182 0.90 POLB (0.46) HCRTR1HCRTR2SIGMAR1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed