SCHEMBL5237555

SCHEMBL5237555

O=C(NCCCc1cccc(N2CC3CN(C(=O)c4c(F)cccc4Cl)CC3C2)c1)c1ccc(F)c(F)c1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 3/20 0.40
RORC P51449 4/20 0.39
HCRTR1 O43613 3/20 0.38
HCRTR2 O43614 3/20 0.38
DRD2 P14416 1/20 0.38
ADRA1A P35348 1/20 0.38
DRD3 P35462 1/20 0.38
MAPT P10636 2/20 0.38
SIGMAR1 Q99720 1/20 0.38
TP53 P04637 1/20 0.38
MEN1 O00255 1/20 0.37
MAPK1 P28482 1/20 0.37
KMT2A Q03164 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
KDM1A O60341 1/20 0.36
HTR1A P08908 1/20 0.36
PLD1 Q13393 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5235222 0.95 HTR1A (0.41) NAMPTRORCHCRTR1HCRTR2DRD2
SCHEMBL5231455 0.94 NAMPT (0.40) NAMPTRORCHCRTR1HCRTR2DRD2
SCHEMBL5230652 0.93 NAMPT (0.42) NAMPTRORCHCRTR1HCRTR2DRD2
SCHEMBL5240254 0.93 NPC1 (0.46) NAMPTRORCHCRTR1HCRTR2DRD2
SCHEMBL5239318 0.92 NPC1 (0.43) NAMPTHCRTR1HCRTR2DRD3MAPT
SCHEMBL5230093 0.92 HCRTR1 (0.39) NAMPTRORCHCRTR1HCRTR2SIGMAR1
SCHEMBL5233648 0.92 HCRTR1 (0.42) HCRTR1HCRTR2SIGMAR1TP53NPC1
SCHEMBL5239914 0.91 HCRTR1 (0.42) NAMPTRORCHCRTR1HCRTR2SIGMAR1
SCHEMBL5233573 0.90 HSD17B10 (0.41) NAMPTHCRTR1HCRTR2DRD2DRD3
SCHEMBL5231603 0.90 NAMPT (0.41) NAMPTRORCHCRTR1HCRTR2SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed