SCHEMBL5231256

SCHEMBL5231256

Cc1ccnc(-c2cccc3c2CCCC3)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.47
CCR5 P51681 1/20 0.47
CCR8 P51685 1/20 0.47
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2A Q12879 1/20 0.40
GRIN2B Q13224 1/20 0.40
GRIN2C Q14957 1/20 0.40
GRIN3A Q8TCU5 1/20 0.40
NOS3 P29474 1/20 0.40
NOS1 P29475 1/20 0.40
NOS2 P35228 1/20 0.40
ADRA1D P25100 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40
CYP2A6 P11509 1/20 0.40
BCL2L1 Q07817 1/20 0.39
BAD Q92934 1/20 0.39
PHGDH O43175 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3367025 0.78 NPY5R (0.48) CCR1CCR5CCR8NOS3NOS1
SCHEMBL24118185 0.77 BCL2L1 (0.36) CYP2A6BCL2L1BADALDH1A1NPC1
SCHEMBL5691234 0.74 NPY5R (0.51) CCR1CCR5CCR8ADRA1ACYP2A6
SCHEMBL9905481 0.74 BCL2L1 (0.43) BCL2L1BADALDH1A1MEN1KMT2A
SCHEMBL24913524 0.74 CCR1 (0.57) CCR1CCR5CCR8NOS3NOS1
SCHEMBL15345164 0.74 CCR1 (0.49) CCR1CCR5CCR8GRIN2DGRIN3B
SCHEMBL987521 0.73 CCR1 (0.61) CCR1CCR5CCR8ADRA1DADRA1A
Ammonia Solution, Strong SCHEMBL5691104 0.73 NPY5R (0.50) CCR1CCR5CCR8ADRA1ACYP2A6
SCHEMBL3977581 0.73 NPC1 (0.51) CYP2A6BCL2L1BADMEN1KMT2A
SCHEMBL4974372 0.72 BCL2L1 (0.60) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1565443-A4 ACETYL 2-HYDROXY-1,3 DIAMINOALKANES ELAN PHARM INC (US) 2007-07-18 EP disclosed
EP-1565443-A2 ACETYL 2-HYDROXY-1,3 DIAMINOALKANES Elan Pharmaceuticals, Inc. (US) 2005-08-24 EP disclosed
WO-2004024081-A2 ACETYL 2-HYDROXY-1,3 DIAMINOALKANES ELAN PHARMACEUTICALS, INC. (US) 2004-03-25 WO disclosed