SCHEMBL5232157

SCHEMBL5232157

CC(C)c1cccc(C(Cc2ccnc3ccccc23)=NN2CCCC2=O)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 3/20 0.42
TGFBR1 P36897 3/20 0.42
MAPK14 Q16539 3/20 0.42
CYP1A2 P05177 1/20 0.36
LMNA P02545 3/20 0.32
XIAP P98170 1/20 0.32
ADAM17 P78536 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
HIF1A Q16665 1/20 0.32
FAAH O00519 1/20 0.32
ALDH1A1 P00352 3/20 0.31
KDM4E B2RXH2 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
MKNK1 Q9BUB5 1/20 0.31
MKNK2 Q9HBH9 1/20 0.31
RAB9A P51151 1/20 0.31
PDE4A P27815 1/20 0.31
LOXL2 Q9Y4K0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5232151 1.00 THRB (0.42) THRBTGFBR1MAPK14CYP1A2LMNA
SCHEMBL5240531 0.88 CYP1A2 (0.38) THRBTGFBR1MAPK14CYP1A2LMNA
SCHEMBL5240528 0.88 CYP1A2 (0.38) THRBTGFBR1MAPK14CYP1A2LMNA
SCHEMBL5234868 0.88 TGFBR1 (0.39) THRBTGFBR1MAPK14CYP1A2LMNA
SCHEMBL5234860 0.88 TGFBR1 (0.39) THRBTGFBR1MAPK14CYP1A2LMNA
SCHEMBL5237953 0.86 CYP1A2 (0.38) THRBTGFBR1MAPK14CYP1A2LMNA
SCHEMBL5237961 0.86 CYP1A2 (0.38) THRBTGFBR1MAPK14CYP1A2LMNA
SCHEMBL5234770 0.84 CYP1A2 (0.38) THRBTGFBR1MAPK14CYP1A2LMNA
SCHEMBL5234762 0.84 CYP1A2 (0.38) THRBTGFBR1MAPK14CYP1A2LMNA
SCHEMBL5238471 0.84 PDE4A (0.38) TGFBR1CYP1A2ADAM17FAAHALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397364-B1 NOVEL PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS LILLY CO ELI (US) 2007-07-25 EP disclosed