SCHEMBL5232170

SCHEMBL5232170

COC(=O)c1ccc(CC(NC(=O)OC(C)(C)C)c2ccc(C(=O)O)cc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.46
ALDH1A1 P00352 3/20 0.45
LMNA P02545 2/20 0.45
PKM P14618 2/20 0.45
HPGD P15428 2/20 0.45
TSHR P16473 2/20 0.45
HTT P42858 2/20 0.45
NPSR1 Q6W5P4 2/20 0.45
HSD17B10 Q99714 2/20 0.45
TP53 P04637 1/20 0.45
MAPT P10636 1/20 0.45
AGTR1 P30556 1/20 0.45
RAB9A P51151 1/20 0.45
CTSS P25774 6/20 0.42
CTSK P43235 5/20 0.42
MEN1 O00255 1/20 0.42
ALOX15 P16050 1/20 0.42
XBP1 P17861 1/20 0.42
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6630454 1.00 ATM (0.46) ATMALDH1A1LMNAPKMHPGD
SCHEMBL5151480 0.95 ATM (0.46) ATMALDH1A1LMNAPKMHPGD
SCHEMBL14588990 0.92 ATM (0.52) ATMALDH1A1LMNAPKMHPGD
SCHEMBL2791088 0.83 ATM (0.41) ATMTSHRMAPTCTSSCTSK
SCHEMBL30109148 0.82 RIPK1 (0.42) ATMTSHRMAPTCTSSCTSK
SCHEMBL989453 0.82 RIPK1 (0.42) ATMTSHRMAPTCTSSCTSK
SCHEMBL31269567 0.81 LOXL2 (0.45) ATMTSHRMAPTCTSSCTSK
SCHEMBL30109275 0.81 LOXL2 (0.45) ATMTSHRMAPTCTSSCTSK
SCHEMBL31269590 0.81 CYP3A4 (0.40) ATMTSHRMAPTCTSSCTSK
SCHEMBL5155482 0.81 NAMPT (0.47) ATMALDH1A1LMNAPKMHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1373233-B1 DERIVATIVES OF N-(ARYLSULFONYL)BETA-AMINOACIDS COMPRISING A SUBSTITUTED AMINOMETHYL GROUP, THE PREPARATION METHOD THEREOF AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SANOFI AVENTIS (FR) 2007-09-05 EP disclosed
EP-1373233-A1 DERIVATIVES OF N-(ARYLSULFONYL)BETA-AMINOACIDS COMPRISING A SUBSTITUTED AMINOMETHYL GROUP, THE PREPARATION METHOD THEREOF AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING SAME Sanofi-Aventis (FR) 2004-01-02 EP disclosed
WO-2002076964-A1 DERIVATIVES OF N-(ARYLSULFONYL)BETA-AMINOACIDS COMPRISING A SUBSTITUTED AMINOMETHYL GROUP, THE PREPARATION METHOD THEREOF AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SANOFI-SYNTHELABO (FR) 2002-10-03 WO disclosed