SCHEMBL5232895

SCHEMBL5232895

COc1ccc(CCCC(N)=O)cc1N1CC2CN(C(=O)c3c(C)cccc3C)CC2C1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 18/20 0.47
HCRTR2 O43614 18/20 0.47
KCNH2 Q12809 1/20 0.41
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5231170 0.82 HCRTR1 (0.52) HCRTR1HCRTR2KCNH2
SCHEMBL4692413 0.77 HCRTR1 (0.53) HCRTR1HCRTR2KCNH2
SCHEMBL5238954 0.74 HCRTR1 (0.43) HCRTR1HCRTR2KMT2A
SCHEMBL5235460 0.73 HCRTR1 (0.50) HCRTR1HCRTR2KCNH2
SCHEMBL5236364 0.72 HCRTR1 (0.47) HCRTR1HCRTR2KCNH2
SCHEMBL4696789 0.71 CCR5 (0.57) HCRTR1HCRTR2KCNH2
SCHEMBL5237889 0.71 HCRTR1 (0.53) HCRTR1HCRTR2KCNH2
SCHEMBL5230893 0.71 HCRTR1 (0.41) HCRTR1HCRTR2KCNH2
SCHEMBL5237741 0.70 HCRTR1 (0.44) HCRTR1HCRTR2KCNH2
SCHEMBL4698184 0.69 HCRTR1 (0.46) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP disclosed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO disclosed