SCHEMBL5233146

SCHEMBL5233146

CC(C)(C)OC(=O)C1CC[C@H](NCCc2ccccc2)C(C(=O)O)C1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
MAPT P10636 2/20 0.46
KDM4E B2RXH2 1/20 0.46
FUCA1 P04066 4/20 0.44
TAAR1 Q96RJ0 6/20 0.43
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39
KMT2A Q03164 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MEN1 O00255 1/20 0.37
RECQL P46063 1/20 0.37
MGAM O43451 1/20 0.37
SI P14410 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
STS P08842 1/20 0.37
GRM2 Q14416 1/20 0.37
GRM3 Q14832 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5029374 0.77 ALDH1A1 (0.44) ALDH1A1GAANPC1RAB9A
SCHEMBL5233189 0.76 RECQL (0.40) TAAR1POLBGAAL3MBTL1RECQL
SCHEMBL5033798 0.76 RECQL (0.40) TAAR1POLBGAAL3MBTL1RECQL
SCHEMBL3641064 0.73 TAAR1 (0.65) ALDH1A1MAPTKDM4ETAAR1POLB
SCHEMBL991353 0.73 TAAR1 (0.65) ALDH1A1MAPTKDM4ETAAR1POLB
SCHEMBL991352 0.73 TAAR1 (0.65) ALDH1A1MAPTKDM4ETAAR1POLB
SCHEMBL6021781 0.72 GPR119 (0.48) ALDH1A1MAPTKDM4EPOLBGAA
SCHEMBL6021777 0.72 GPR119 (0.48) ALDH1A1MAPTKDM4EPOLBGAA
Hydrochloric Acid SCHEMBL993335 0.72 TAAR1 (0.63) ALDH1A1MAPTKDM4ETAAR1POLB
Hydrochloric Acid SCHEMBL993334 0.72 TAAR1 (0.63) ALDH1A1MAPTKDM4ETAAR1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656138-A4 SUBSTITUTED CYCLOALKYAMINE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL MYERS SQUIBB CO (US) 2007-04-18 EP disclosed
EP-1656138-A2 SUBSTITUTED CYCLOALKYAMINE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Bristol-Myers Squibb Company (US) 2006-05-17 EP disclosed
WO-2005020899-A2 SUBSTITUTED CYCLOALKYAMINE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL-MYERS SQUIBB COMPANY (US) 2005-03-10 WO disclosed