SCHEMBL5234520

SCHEMBL5234520

CN(C)C=C1CCN(C(=O)c2ccc([N+](=O)[O-])cc2)c2ccsc2C1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
STING1 Q86WV6 1/20 0.38
MAPT P10636 5/20 0.37
MAPK1 P28482 1/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37
CA14 Q9ULX7 1/20 0.37
LMNA P02545 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
HPGD P15428 2/20 0.36
AVPR2 P30518 1/20 0.36
AVPR1A P37288 1/20 0.36
ATM Q13315 1/20 0.35
BCHE P06276 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5235254 1.00 ALDH1A1 (0.40) ALDH1A1SMN1; SMN2STING1MAPTMAPK1
SCHEMBL5233480 0.85 KMT2A (0.39) ALDH1A1SMN1; SMN2MAPTCA2LMNA
SCHEMBL5233477 0.85 KMT2A (0.39) ALDH1A1SMN1; SMN2MAPTCA2LMNA
SCHEMBL5231836 0.85 STING1 (0.38) ALDH1A1SMN1; SMN2STING1MAPTMAPK1
SCHEMBL7313747 0.85 STING1 (0.38) ALDH1A1SMN1; SMN2STING1MAPTMAPK1
SCHEMBL7330866 0.82 ALDH1A1 (0.46) ALDH1A1SMN1; SMN2STING1MAPTLMNA
SCHEMBL7330871 0.82 ALDH1A1 (0.46) ALDH1A1SMN1; SMN2STING1MAPTLMNA
SCHEMBL5238511 0.80 ALDH1A1 (0.39) ALDH1A1SMN1; SMN2STING1MAPTCA12
SCHEMBL5238517 0.80 ALDH1A1 (0.39) ALDH1A1SMN1; SMN2STING1MAPTCA12
SCHEMBL8688564 0.79 KDM4E (0.38) ALDH1A1SMN1; SMN2MAPTMAPK1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0804440-B1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS WYETH CORP (US) 2007-12-19 EP disclosed
US-5719278-A TREATING EXCESS RENAL REABSORPTION OF WATER AMERICAN CYANAMID COMPANY (US) 1998-02-17 US disclosed
WO-1996022295-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS AMERICAN CYANAMID COMPANY (US) 1996-07-25 WO disclosed
US-5532235-A TO TREAT EXCESS RENAL REABSORPTION AMERICAN CYANAMID COMPANY (US) 1996-07-02 US disclosed