SCHEMBL5234567

SCHEMBL5234567

CC(C)N(c1nn(-c2ccc(C=Cc3ccccn3)cc2)cc1OC(=O)O)C(=O)[C@H]1CC[C@H](C)CC1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 2/20 0.35
KDR P35968 2/20 0.31
OPRM1 P35372 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
HTR1A P08908 1/20 0.31
TSHR P16473 1/20 0.31
LMNA P02545 1/20 0.30
RAB9A P51151 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
GLA P06280 1/20 0.30
HPGD P15428 1/20 0.30
PTGS1 P23219 1/20 0.30
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5229947 0.93 TRPM8 (0.32) NR1H4LMNAKDM4EALDH1A1GLA
SCHEMBL5234966 0.93 TRPM8 (0.32) NR1H4LMNAKDM4EALDH1A1GLA
SCHEMBL5236173 0.89 CYP17A1 (0.30)
SCHEMBL5232278 0.89 NR1H4 (0.34) NR1H4KDROPRM1MEN1KMT2A
SCHEMBL5232272 0.89 NR1H4 (0.34) NR1H4KDROPRM1MEN1KMT2A
SCHEMBL5236283 0.87
SCHEMBL5234535 0.87
SCHEMBL5233878 0.87
SCHEMBL5233446 0.86 NPC1 (0.35) MEN1KMT2ATSHRRAB9AKDM4E
SCHEMBL5233366 0.86

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730116-B1 4-CARBOX PYRAZOLE DERIVATES USEFUL AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORP (US) 2007-09-05 EP claimed