SCHEMBL5233446

SCHEMBL5233446

CC(C)N(c1nn(-c2ccccc2)cc1OC(=O)O)C(=O)[C@H]1CC[C@H](C)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.35
RAB9A P51151 3/20 0.35
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
KDM5B Q9UGL1 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
MAPT P10636 1/20 0.32
GAA P10253 1/20 0.32
TSHR P16473 2/20 0.32
UCHL1 P09936 1/20 0.32
KDM4E B2RXH2 1/20 0.32
USP2 O75604 1/20 0.32
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
PKM P14618 1/20 0.32
ALOX15 P16050 1/20 0.32
HTT P42858 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
HSD17B10 Q99714 1/20 0.32
GLA P06280 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5238208 0.94 ALDH1A1 (0.38) NPC1RAB9AKDM5BMAPTKDM4E
SCHEMBL5234466 0.92 APP (0.36) KMT2AMEN1ADORA3GAAALDH1A1
SCHEMBL5236797 0.92
SCHEMBL5236128 0.92 NPC1 (0.34) NPC1RAB9AKMT2AMEN1KDM5B
SCHEMBL5228396 0.92 KMT2A (0.34) KMT2AMEN1TSHRKDM4EUSP2
SCHEMBL5229947 0.92 TRPM8 (0.32) KDM4EALDH1A1GLA
SCHEMBL5234966 0.92 TRPM8 (0.32) KDM4EALDH1A1GLA
SCHEMBL5239459 0.91 KDM4E (0.33) NPC1RAB9AKMT2AMAPTGAA
SCHEMBL5234344 0.91 ESRRA (0.31)
SCHEMBL5231776 0.91 ESRRA (0.32) NPC1RAB9AKMT2AMEN1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730116-B1 4-CARBOX PYRAZOLE DERIVATES USEFUL AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORP (US) 2007-09-05 EP claimed