SCHEMBL5235015

SCHEMBL5235015

NN=C(Cc1ccnc2ccccc12)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 1/20 0.43
CYP1A2 P05177 1/20 0.43
CNR2 P34972 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.38
BCHE P06276 1/20 0.37
FLT1 P17948 2/20 0.37
KDR P35968 2/20 0.37
MCHR1 Q99705 1/20 0.37
GRIN2B Q13224 2/20 0.36
ABCG2 Q9UNQ0 2/20 0.36
TACR1 P25103 1/20 0.36
HDAC3 O15379 1/20 0.36
ACHE P22303 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HDAC9 Q9UKV0 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5237502 1.00 LOXL2 (0.43) LOXL2CYP1A2CNR2PTGDR2BCHE
SCHEMBL5240093 0.87 CNR2 (0.45) LOXL2CYP1A2CNR2FLT1KDR
SCHEMBL5231738 0.87 CNR2 (0.45) LOXL2CYP1A2CNR2FLT1KDR
SCHEMBL5234948 0.86 LOXL2 (0.46) LOXL2CYP1A2HDAC3ACHEHDAC1
SCHEMBL5234952 0.86 LOXL2 (0.46) LOXL2CYP1A2HDAC3ACHEHDAC1
SCHEMBL5238056 0.85 CYP1A2 (0.54) LOXL2CYP1A2HDAC3ACHEHDAC1
SCHEMBL5238727 0.85 CYP1A2 (0.54) LOXL2CYP1A2HDAC3ACHEHDAC1
SCHEMBL5235754 0.85 AURKA (0.39) LOXL2CYP1A2CNR2FLT1KDR
SCHEMBL5235758 0.85 AURKA (0.39) LOXL2CYP1A2CNR2FLT1KDR
SCHEMBL5238458 0.83 LOXL2 (0.46) LOXL2CYP1A2FLT1KDRTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397364-B1 NOVEL PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS LILLY CO ELI (US) 2007-07-25 EP disclosed
CN-1951939-A Novel pyrrole derivatives as pharmaceutical agents LILLY CO ELI (US) 2007-04-25 CN disclosed
CN-1269820-C Novel pyrrole derivatives as medicaments LILLY CO ELI (US) 2006-08-16 CN disclosed
CN-1511157-A Novel pyrrole derivatives as medicaments 2004-07-07 CN disclosed