SCHEMBL5236444

SCHEMBL5236444

O=CCc1c(Br)ccc2ccccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 5/20 0.40
CYP1A2 P05177 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
ALDH1A1 P00352 5/20 0.39
TDP1 Q9NUW8 2/20 0.39
CYP2A6 P11509 1/20 0.39
TSHR P16473 1/20 0.39
KDM4E B2RXH2 4/20 0.39
GAA P10253 3/20 0.39
GLA P06280 1/20 0.39
HPGD P15428 1/20 0.39
MAPT P10636 3/20 0.38
TAAR1 Q96RJ0 1/20 0.38
ERN1 O75460 1/20 0.38
POLB P06746 1/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6620341 0.82 HSD17B10 (0.38) HSD17B10CYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL7924281 0.81 HSD17B10 (0.40) HSD17B10CYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL15351705 0.79 ALDH1A1 (0.44) HSD17B10CYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL2467403 0.78 HSD17B10 (0.63) HSD17B10CYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL3414797 0.78 CYP2A6 (0.48) HSD17B10CYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL9404144 0.76 HTR2A (0.54) HSD17B10CYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL8988212 0.76 ALDH1A1 (0.46) HSD17B10CYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL7783948 0.75 NCEH1 (0.45) HSD17B10CYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL18070730 0.75 ALDH1A1 (0.44) HSD17B10CYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL6403906 0.75 ALDH1A1 (0.60) HSD17B10CYP1A2CYP2C9CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118772148-A Imidazo [1,2-a ] pyrimidine matrine/sophoridine derivative, preparation method and application 西北农林科技大学 2024-10-15 CN disclosed
EP-3322705-A1 2-AMINO-1,3,4-THIADIAZINE AND 2-AMINO-1,3,4-OXADIAZINE BASED ANTIFUNGAL AGENTS F2G Limited (GB) 2018-05-23 EP disclosed
WO-2017009651-A1 2-AMINO-1,3,4-THIADIAZINE AND 2-AMINO-1,3,4-OXADIAZINE BASED ANTIFUNGAL AGENTS F2G LIMITED (GB) 2017-01-19 WO disclosed
EP-1851232-A2 DIHYDROIMIDAZOTHIAZOLE DERIVATIVES Prosidion Limited (GB) 2007-11-07 EP disclosed
WO-2006085118-A2 DIHYDROIMIDAZOTHIAZOLE DERIVATIVES PROSIDION LIMITED (GB) 2006-08-17 WO disclosed
EP-1474140-A1 2-OXAZOLAMINES AND THEIR USE AS 5-HT2B RECEPTOR ANTAGONISTS Pharmagene Laboratories Ltd (GB) 2004-11-10 EP disclosed
WO-2003068226-A1 2-OXAZOLAMINES AND THEIR USE AS 5-HT2B RECEPTOR ANTAGONISTS PHARMAGENE LABORATORIES LIMITED (GB) 2003-08-21 WO disclosed