SCHEMBL5237627

SCHEMBL5237627

O=C(O)Oc1cc2cc(F)cc(F)c2s1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 1/20 0.36
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
GAA P10253 4/20 0.33
KMT2A Q03164 2/20 0.33
ERN1 O75460 1/20 0.32
LMNA P02545 2/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
NOTUM Q6P988 1/20 0.31
AKR1B1 P15121 2/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
TNF P01375 1/20 0.30
MAPT P10636 1/20 0.30
HPGD P15428 1/20 0.30
HTT P42858 1/20 0.30
MCL1 Q07820 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
NOD2 Q9HC29 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5230123 0.83 CHRNA7 (0.38) CHRNA7CES2CES1GAAKMT2A
SCHEMBL5233818 0.79 CHRNA7 (0.39) CHRNA7CES2CES1GAANPC1
SCHEMBL2898184 0.74 GPR35 (0.48) CHRNA7CES2CES1KMT2ANOTUM
SCHEMBL5234254 0.74 KMT2A (0.39) CHRNA7KMT2ALMNANPC1RAB9A
SCHEMBL2892797 0.72 CHRNA7 (0.46) CHRNA7GAAKMT2ALMNANPC1
SCHEMBL5238184 0.70 KMT2A (0.41) CHRNA7GAAKMT2ALMNAMEN1
SCHEMBL19546521 0.70 CES2 (0.41) CES2CES1GAAKMT2AERN1
SCHEMBL12490192 0.68 CLK1 (0.51) CHRNA7LMNAMAPT
SCHEMBL12490653 0.68 CYP2A6 (0.41) CHRNA7ERN1RAB9ASMN1; SMN2
SCHEMBL1365999 0.68 CES2 (0.37) CHRNA7CES2CES1ERN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1461335-B1 2-HETEROARYLCARBOXYLIC ACID AMIDES BAYER HEALTHCARE AG (DE) 2007-02-28 EP disclosed
EP-1461335-A1 2-HETEROARYLCARBOXYLIC ACID AMIDES Bayer HealthCare AG (DE) 2004-09-29 EP disclosed
WO-2003055878-A1 2-HETEROARYLCARBOXYLIC ACID AMIDES BAYER HEALTHCARE AG (DE) 2003-07-10 WO disclosed