SCHEMBL5237789

SCHEMBL5237789

Cc1ncnc(C)c1C(=O)N1CC2CN(CCC(NC(=O)C3CCC(F)(F)CC3)c3cccc(F)c3)C[C@H]2C1

nearest known ligand 0.81

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 18/20 0.81
CCL5 P13501 4/20 0.60
KCNH2 Q12809 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13326712 1.00 CCR5 (0.81) CCR5CCL5KCNH2
SCHEMBL30227416 0.92 CCR5 (0.80) CCR5CCL5KCNH2
SCHEMBL5422017 0.91 CCR5 (0.82) CCR5
SCHEMBL13326700 0.91 CCR5 (0.82) CCR5
Cyclopentane SCHEMBL4693960 0.86 CCR5 (0.80) CCR5CCL5KCNH2
SCHEMBL4978839 0.85 CCR5 (0.65) CCR5CCL5KCNH2
SCHEMBL30227485 0.85 CCR5 (0.73) CCR5CCL5KCNH2
SCHEMBL30227516 0.84 CCR5 (0.68) CCR5
SCHEMBL14448125 0.82 CCR5 (0.72) CCR5CCL5KCNH2
SCHEMBL13326710 0.82 CCR5 (0.72) CCR5CCL5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed