SCHEMBL5237932

SCHEMBL5237932

CCCc1cccc(C(=O)Cc2ccnc3ccccc23)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.48
KDM4E B2RXH2 2/20 0.43
LOXL2 Q9Y4K0 1/20 0.39
PDE4A P27815 1/20 0.38
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
GAA P10253 1/20 0.36
PDE10A Q9Y233 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
GLS O94925 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
HTR1A P08908 1/20 0.35
ADRA1D P25100 1/20 0.35
ADRA1A P35348 1/20 0.35
ADRA1B P35368 1/20 0.35
FERMT2 Q96AC1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29959944 0.90 CYP1A2 (0.47) CYP1A2LOXL2PDE4AMEN1KMT2A
SCHEMBL5234356 0.90 CYP1A2 (0.47) CYP1A2LOXL2PDE4AMEN1KMT2A
SCHEMBL5235225 0.82 CYP1A2 (0.49) CYP1A2LOXL2PDE4AALDH1A1SMN1; SMN2
SCHEMBL29959459 0.82 CYP1A2 (0.49) CYP1A2LOXL2PDE4AALDH1A1SMN1; SMN2
SCHEMBL5233274 0.82 CYP1A2 (0.55) CYP1A2KDM4ELOXL2PDE4AALDH1A1
SCHEMBL5236988 0.80 CYP1A2 (0.49) CYP1A2KDM4ELOXL2PDE4AALDH1A1
SCHEMBL5236887 0.80 CYP1A2 (0.49) CYP1A2KDM4ELOXL2PDE4AALDH1A1
SCHEMBL4872415 0.80 CYP1A2 (0.49) CYP1A2KDM4ELOXL2PDE4AALDH1A1
SCHEMBL5235242 0.79 CYP1A2 (0.46) CYP1A2LOXL2PDE4AMEN1KMT2A
SCHEMBL4872056 0.77 CYP1A2 (0.55) CYP1A2KDM4ELOXL2KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397364-B1 NOVEL PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS LILLY CO ELI (US) 2007-07-25 EP disclosed