SCHEMBL5238484

SCHEMBL5238484

CCCCOc1c(CNC(=O)O)n(CCC(=O)NC(C)C)c(=O)c2cc(Cl)c(Cl)cc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.37
NLRP1 Q9C000 1/20 0.37
PLK1 P53350 3/20 0.37
AVPR1B P47901 3/20 0.36
CNR2 P34972 1/20 0.36
TP53 P04637 1/20 0.35
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
TSHR P16473 1/20 0.34
CYP3A4 P08684 2/20 0.33
CYP2C9 P11712 2/20 0.33
MAPT P10636 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33
MEN1 O00255 1/20 0.33
PKM P14618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5239739 0.87 HPGD (0.39) HPGDNLRP1PLK1AVPR1BCNR2
SCHEMBL5238212 0.87 RXFP1 (0.34) CNR2TP53ALDH1A1GAAMAPT
SCHEMBL5235009 0.86 DPP4 (0.38) ALDH1A1
SCHEMBL5236293 0.85 ALDH1A1 (0.41) HPGDCNR2TP53KDM4EALDH1A1
SCHEMBL6704499 0.85 PTGER4 (0.33) AVPR1BCNR2
SCHEMBL6107675 0.84 HPGD (0.35) HPGDNLRP1PLK1AVPR1BCNR2
SCHEMBL6703529 0.83 DPP4 (0.35) KDM4EKMT2A
SCHEMBL5238488 0.82 HPGD (0.37) HPGDNLRP1PLK1AVPR1BCNR2
SCHEMBL5234470 0.81 THRA (0.36) HPGDCNR2ALDH1A1HTTSMN1; SMN2
SCHEMBL5236977 0.81 SMN1; SMN2 (0.34) HPGDCNR2KDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1355886-B1 FUSED HETEROCYCLIC COMPOUNDS TAKEDA PHARMACEUTICAL (JP) 2007-07-11 EP disclosed