SCHEMBL5239559

SCHEMBL5239559

O=C(Cc1ccnc2ccccc12)c1cccc(OC(F)(F)F)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KAT6A Q92794 3/20 0.44
KDR P35968 2/20 0.44
RAF1 P04049 1/20 0.44
LCK P06239 1/20 0.44
RET P07949 1/20 0.44
CYP3A4 P08684 1/20 0.44
KIT P10721 1/20 0.44
MAP3K20 Q9NYL2 1/20 0.44
RIPK3 Q9Y572 1/20 0.44
TRPV1 Q8NER1 2/20 0.44
CYP1A2 P05177 1/20 0.43
MGLL Q99685 1/20 0.43
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
BRAF P15056 3/20 0.40
MAPK14 Q16539 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
TNNI3K Q59H18 1/20 0.39
TAS1R3 Q7RTX0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5232145 0.83 RAF1 (0.40) KAT6AKDRRAF1LCKRET
SCHEMBL5232140 0.83 RAF1 (0.40) KAT6AKDRRAF1LCKRET
SCHEMBL5233508 0.82 CNR2 (0.53) KDRCYP1A2BRAFMAPK14TNNI3K
SCHEMBL5231753 0.80 CYP1A2 (0.53) CYP3A4CYP1A2MEN1KMT2A
SCHEMBL29987166 0.78 CYP1A2 (0.61) CYP3A4CYP1A2MEN1KMT2A
SCHEMBL5239658 0.78 CYP1A2 (0.61) CYP3A4CYP1A2MEN1KMT2A
SCHEMBL5234876 0.78 CYP1A2 (0.49) KDRCYP1A2MEN1KMT2A
SCHEMBL27515586 0.77 TRPV1 (0.45) KDRRAF1LCKRETCYP3A4
SCHEMBL5238033 0.77 MGLL (0.41) KDRRAF1LCKRETCYP3A4
SCHEMBL5238037 0.77 MGLL (0.41) KDRRAF1LCKRETCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397364-B1 NOVEL PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS LILLY CO ELI (US) 2007-07-25 EP disclosed