SCHEMBL5234876

SCHEMBL5234876

O=C(Cc1ccnc2ccccc12)c1cccc(Cl)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.49
PSMD14 O00487 1/20 0.48
NPC1 O15118 1/20 0.48
MAPK1 P28482 1/20 0.48
RAB9A P51151 1/20 0.48
CTDSP1 Q9GZU7 1/20 0.48
TACR1 P25103 1/20 0.46
FADS1 O60427 1/20 0.46
ERCC5 P28715 1/20 0.44
FEN1 P39748 1/20 0.44
LOXL2 Q9Y4K0 1/20 0.43
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 1/20 0.42
GLA P06280 1/20 0.42
CTSV O60911 1/20 0.41
CTSL P07711 1/20 0.41
CTSS P25774 1/20 0.41
FLT1 P17948 1/20 0.41
KDR P35968 1/20 0.41
PARP1 P09874 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5233678 0.85 RAB9A (0.56) CYP1A2NPC1MAPK1RAB9ATACR1
SCHEMBL29987166 0.84 CYP1A2 (0.61) CYP1A2NPC1MAPK1RAB9ALOXL2
SCHEMBL5239658 0.84 CYP1A2 (0.61) CYP1A2NPC1MAPK1RAB9ALOXL2
SCHEMBL5231753 0.84 CYP1A2 (0.53) CYP1A2NPC1RAB9ALOXL2KDM4E
SCHEMBL5233929 0.82 CYP1A2 (0.50) CYP1A2PSMD14NPC1MAPK1RAB9A
SCHEMBL5241399 0.81 FADS1 (0.46) CYP1A2PSMD14NPC1MAPK1RAB9A
SCHEMBL5241402 0.81 FADS1 (0.46) CYP1A2PSMD14NPC1MAPK1RAB9A
SCHEMBL5233508 0.81 CNR2 (0.53) CYP1A2NPC1RAB9AALDH1A1FLT1
SCHEMBL9033128 0.78 NPC1 (0.50) PSMD14NPC1MAPK1RAB9ACTDSP1
SCHEMBL5239559 0.78 KAT6A (0.44) CYP1A2KDRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397364-B1 NOVEL PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS LILLY CO ELI (US) 2007-07-25 EP disclosed