SCHEMBL5239698

SCHEMBL5239698

O=C1CCCN1N=C(Cc1ccnc2ccccc12)c1cccc(C(F)(F)F)c1F

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.38
CYP1A2 P05177 1/20 0.35
TRPV1 Q8NER1 1/20 0.35
AURKA O14965 2/20 0.35
AURKB Q96GD4 1/20 0.35
P2RX7 Q99572 10/20 0.35
DGAT2 Q96PD7 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5238769 0.86 CYP1A2 (0.40) KDRCYP1A2
SCHEMBL5238764 0.86 CYP1A2 (0.40) KDRCYP1A2
SCHEMBL5238619 0.83 KDR (0.35) KDRCYP1A2AURKA
SCHEMBL5233924 0.81 KDR (0.38) KDRCYP1A2DGAT2
SCHEMBL5233927 0.81 KDR (0.38) KDRCYP1A2DGAT2
SCHEMBL5235220 0.81 KDR (0.44) KDRCYP1A2DGAT2POLB
SCHEMBL5235216 0.81 KDR (0.44) KDRCYP1A2DGAT2POLB
SCHEMBL5235150 0.80 CYP1A2 (0.40) CYP1A2
SCHEMBL5235146 0.80 CYP1A2 (0.40) CYP1A2
SCHEMBL5239587 0.79 AR (0.39) KDRCYP1A2P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397364-B1 NOVEL PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS LILLY CO ELI (US) 2007-07-25 EP disclosed