SCHEMBL5243082

SCHEMBL5243082

CCCCc1c(C#N)sc2nc3c(cc12)CCCC3

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 13/20 0.60
ALDH1A1 P00352 8/20 0.60
MAPT P10636 7/20 0.60
LMNA P02545 5/20 0.60
SMN1; SMN2 Q16637 10/20 0.48
HSD17B10 Q99714 5/20 0.48
HPGD P15428 4/20 0.48
HTT P42858 3/20 0.48
MAPK1 P28482 2/20 0.48
NPSR1 Q6W5P4 2/20 0.48
TSHR P16473 2/20 0.48
L3MBTL1 Q9Y468 2/20 0.43
ALOX15 P16050 1/20 0.43
RAB9A P51151 7/20 0.41
NPC1 O15118 6/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
POLB P06746 3/20 0.39
EEF2K O00418 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4703593 0.78 NPC1 (0.51) KDM4EALDH1A1MAPTLMNASMN1; SMN2
SCHEMBL4705357 0.77 NPC1 (0.50) KDM4EALDH1A1MAPTLMNASMN1; SMN2
SCHEMBL5243084 0.76 KDM4E (0.43) KDM4EALDH1A1MAPTLMNASMN1; SMN2
SCHEMBL4703597 0.66 ALDH1A1 (0.40) KDM4EALDH1A1MAPTLMNASMN1; SMN2
SCHEMBL13154828 0.66 KDM4E (0.63) KDM4EALDH1A1MAPTLMNASMN1; SMN2
SCHEMBL14954867 0.62 MAPT (0.64) KDM4EALDH1A1MAPTLMNASMN1; SMN2
SCHEMBL13154843 0.61 KDM4E (0.65) KDM4EALDH1A1MAPTLMNASMN1; SMN2
SCHEMBL15116256 0.61 SMN1; SMN2 (0.65) KDM4EALDH1A1SMN1; SMN2HSD17B10HTT
SCHEMBL23378351 0.61 NPC1 (0.77) KDM4EALDH1A1MAPTLMNASMN1; SMN2
SCHEMBL8388800 0.61 SMN1; SMN2 (0.59) KDM4EALDH1A1LMNASMN1; SMN2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863571-A1 COMPOUNDS FOR INHIBITING KSP KINESIN ACTIVITY Shering Corporation (US) 2007-12-12 EP disclosed
WO-2006098962-A1 COMPOUNDS FOR INHIBITING KSP KINESIN ACTIVITY SCHERING CORPORATION (US) 2006-09-21 WO disclosed