SCHEMBL5243274

SCHEMBL5243274

Nc1[nH]c2sc3c(N)ncnc3c2c2cccc1-2

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LIMK1 P53667 17/20 0.52
CDC7 O00311 5/20 0.46
CDK5 Q00535 2/20 0.46
PLK4 O00444 2/20 0.46
AURKA O14965 2/20 0.46
ROCK2 O75116 2/20 0.46
PIM1 P11309 2/20 0.46
PRKACA P17612 2/20 0.46
RPS6KB1 P23443 2/20 0.46
CDK2 P24941 2/20 0.46
MARK3 P27448 2/20 0.46
FLT4 P35916 2/20 0.46
KDR P35968 2/20 0.46
CSNK1D P48730 2/20 0.46
GSK3A P49840 2/20 0.46
STK3 Q13188 2/20 0.46
ROCK1 Q13464 2/20 0.46
DYRK1A Q13627 2/20 0.46
MARK2 Q7KZI7 2/20 0.46
AURKB Q96GD4 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5244491 0.79 LIMK1 (0.61) LIMK1CDC7CDK5PLK4AURKA
SCHEMBL5243145 0.76 LIMK1 (0.34) LIMK1
SCHEMBL12822244 0.69 LIMK1 (1.00) LIMK1CDC7CDK5PLK4AURKA
SCHEMBL12969821 0.65 LIMK1 (0.76) LIMK1CDK5KDRMAP4K4CDK5R1
SCHEMBL12969829 0.65 LIMK1 (0.72) LIMK1CDC7CDK5PLK4AURKA
SCHEMBL12970350 0.65 LIMK1 (0.76) LIMK1CDC7CDK5PLK4AURKA
SCHEMBL4896988 0.65 IDO1 (0.46) LIMK1CDC7CDK5PIM1DYRK1A
SCHEMBL12969561 0.65 LIMK1 (0.56) LIMK1CDK5CDK5R1CLK1
SCHEMBL12969576 0.64 LIMK1 (1.00) LIMK1CDC7CDK5CDK5R1CLK1
SCHEMBL12969575 0.63 LIMK1 (0.71) LIMK1CDK5CDK5R1CLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1819710-A1 NEW PYRIDOTHIENOPYRIMIDINE DERIVATIVES Laboratorios Almirall, S.A. (ES) 2007-08-22 EP claimed
WO-2006058724-A1 NEW PYRIDOTHIENOPYRIMIDINE DERIVATIVES LABORATORIOS ALMIRALL, S.A. (ES) 2006-06-08 WO claimed
EP-1819710-A1 NEW PYRIDOTHIENOPYRIMIDINE DERIVATIVES Laboratorios Almirall, S.A. (ES) 2007-08-22 EP disclosed
WO-2006058724-A1 NEW PYRIDOTHIENOPYRIMIDINE DERIVATIVES LABORATORIOS ALMIRALL, S.A. (ES) 2006-06-08 WO disclosed