SCHEMBL5244307

SCHEMBL5244307

O=C(NCC(F)(F)F)c1ccc(-n2cc(C(=O)NCc3cccc(C(F)(F)F)c3)nn2)c(OCCOCCF)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DDT P30046 3/20 0.50
PSEN1 P49768 1/20 0.50
PSEN2 P49810 1/20 0.50
APH1B Q8WW43 1/20 0.50
NCSTN Q92542 1/20 0.50
APH1A Q96BI3 1/20 0.50
PSENEN Q9NZ42 1/20 0.50
MLYCD O95822 1/20 0.43
ROCK2 O75116 1/20 0.42
ROCK1 Q13464 1/20 0.42
MAPK14 Q16539 1/20 0.42
MMP13 P45452 3/20 0.42
GLS O94925 6/20 0.42
MEN1 O00255 1/20 0.41
PLA2G1B P04054 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
GAA P10253 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5246799 0.93 PSEN1 (0.41) DDTPSEN1PSEN2APH1BNCSTN
SCHEMBL5244424 0.93 DDT (0.52) DDTPSEN1PSEN2APH1BNCSTN
SCHEMBL3111267 0.92 GLS (0.43) DDTPSEN1PSEN2APH1BNCSTN
SCHEMBL5246995 0.92 DDT (0.41) DDTPSEN1PSEN2APH1BNCSTN
SCHEMBL5246041 0.92 MIF (0.45) DDTPSEN1PSEN2APH1BNCSTN
SCHEMBL5250510 0.91 DDT (0.41) DDTPSEN1PSEN2APH1BNCSTN
SCHEMBL5248520 0.91 DDT (0.41) DDTPSEN1PSEN2APH1BNCSTN
SCHEMBL5248368 0.90 NAMPT (0.40) DDTPSEN1PSEN2APH1BNCSTN
SCHEMBL5244881 0.90 GLS (0.49) ROCK2ROCK1MAPK14GLS
SCHEMBL5247215 0.90 DDT (0.46) DDTPSEN1PSEN2APH1BNCSTN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1867331-A1 TRIAZOLE DERIVATIVE AND THE USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-12-19 EP disclosed