SCHEMBL5246995

SCHEMBL5246995

O=C(NCC(F)(F)F)c1ccc(-n2cc(C(=O)NCc3ccc(C(F)(F)F)cc3)nn2)c(OCCOCCF)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DDT P30046 3/20 0.41
KDM1A O60341 2/20 0.40
HDAC1 Q13547 2/20 0.40
PSEN1 P49768 1/20 0.40
PSEN2 P49810 1/20 0.40
APH1B Q8WW43 1/20 0.40
NCSTN Q92542 1/20 0.40
APH1A Q96BI3 1/20 0.40
PSENEN Q9NZ42 1/20 0.40
MIF P14174 1/20 0.39
MAPK14 Q16539 1/20 0.38
MMP13 P45452 1/20 0.38
GLS O94925 1/20 0.38
LSS P48449 1/20 0.38
DRD2 P14416 1/20 0.37
ROCK2 O75116 1/20 0.37
EPHX2 P34913 1/20 0.37
NAMPT P43490 1/20 0.36
PPARG P37231 1/20 0.36
PPARD Q03181 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5247166 0.94 EPHX2 (0.41) DDTMIFEPHX2
SCHEMBL5246799 0.94 PSEN1 (0.41) DDTPSEN1PSEN2APH1BNCSTN
SCHEMBL5246077 0.93 MMP13 (0.37) DDTPSEN1PSEN2APH1BNCSTN
SCHEMBL5247395 0.92 DDT (0.43) DDTKDM1AHDAC1PSEN1PSEN2
SCHEMBL5246041 0.92 MIF (0.45) DDTPSEN1PSEN2APH1BNCSTN
SCHEMBL5244307 0.92 DDT (0.50) DDTPSEN1PSEN2APH1BNCSTN
SCHEMBL5248368 0.91 NAMPT (0.40) DDTPSEN1PSEN2APH1BNCSTN
SCHEMBL5244132 0.91 HTR2C (0.43) GLSEPHX2NAMPTPPARGPPARA
SCHEMBL5248109 0.91 EGLN1 (0.38) DDTPSEN1PSEN2APH1BNCSTN
Trifluoroacetic Acid SCHEMBL5244494 0.90 MIF (0.37) DDTMIFMAPK14MMP13GLS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1867331-A1 TRIAZOLE DERIVATIVE AND THE USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-12-19 EP disclosed