SCHEMBL5246258

SCHEMBL5246258

CCNC(=O)c1ccc(-n2cc(C(=O)NCc3ccc(S(C)(=O)=O)cc3)nn2)c(OCCCCCCF)c1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 3/20 0.43
RORC P51449 5/20 0.42
DRD2 P14416 1/20 0.40
MAPK8 P45983 9/20 0.39
MAPK9 P45984 7/20 0.39
MAPK10 P53779 6/20 0.39
PRKD3 O94806 2/20 0.39
MAPK1 P28482 2/20 0.39
PRKD2 Q9BZL6 2/20 0.39
DYRK3 O43781 1/20 0.39
JUN P05412 1/20 0.39
CSF1R P07333 1/20 0.39
RPS27 P42677 1/20 0.39
NR1H4 Q96RI1 1/20 0.39
MIF P14174 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5246284 0.92 EPHX2 (0.49) EPHX2RORCDRD2MAPK8MAPK9
SCHEMBL5244275 0.89 MAPK8 (0.47) EPHX2RORCDRD2MAPK8MAPK9
SCHEMBL5245729 0.86 SMPD1 (0.40)
SCHEMBL5247632 0.85 GLS (0.42) MIF
SCHEMBL3112251 0.84 EPHX2 (0.36) EPHX2NR1H4MIF
SCHEMBL5247900 0.84 SMPD1 (0.44) DRD2
SCHEMBL5244569 0.83 SMPD1 (0.41)
SCHEMBL5247618 0.83 SMPD1 (0.43) DRD2
SCHEMBL5248314 0.83 SMPD1 (0.39)
SCHEMBL5247392 0.83 GLS (0.47) DRD2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1867331-A1 TRIAZOLE DERIVATIVE AND THE USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-12-19 EP disclosed