SCHEMBL5247632

SCHEMBL5247632

CCNC(=O)c1ccc(-n2cc(C(=O)NCc3cccc(F)c3)nn2)c(OCCCCCCF)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLS O94925 1/20 0.42
ROCK2 O75116 2/20 0.42
ROCK1 Q13464 1/20 0.42
CNR1 P21554 1/20 0.42
POLB P06746 1/20 0.41
DDT P30046 2/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
MMP13 P45452 1/20 0.40
BRD4 O60885 2/20 0.40
PSEN1 P49768 2/20 0.40
PSEN2 P49810 2/20 0.40
APH1B Q8WW43 2/20 0.40
NCSTN Q92542 2/20 0.40
APH1A Q96BI3 2/20 0.40
PSENEN Q9NZ42 2/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
PDE10A Q9Y233 1/20 0.39
MIF P14174 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5246709 0.92 ROCK2 (0.42) GLSROCK2ROCK1CNR1POLB
SCHEMBL5247715 0.91 GLS (0.45) GLSROCK2ROCK1CNR1POLB
SCHEMBL5246018 0.89 POLB (0.42) GLSROCK2ROCK1CNR1POLB
SCHEMBL5244706 0.85 ROCK2 (0.40) ROCK2ROCK1DDTBRD4PSEN1
SCHEMBL5246258 0.85 EPHX2 (0.43) MIF
SCHEMBL5246108 0.85 BRD4 (0.47) POLBMAPTBRD4
SCHEMBL5247392 0.85 GLS (0.47) GLSROCK2ROCK1POLBBRD4
SCHEMBL5246401 0.85 BRD4 (0.41) POLBMAPTBRD4PSEN1PSEN2
SCHEMBL3112251 0.85 EPHX2 (0.36) ROCK2ROCK1DDTBRD4PSEN1
SCHEMBL5247900 0.84 SMPD1 (0.44) BRD4TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1867331-A1 TRIAZOLE DERIVATIVE AND THE USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-12-19 EP disclosed