SCHEMBL5246346

SCHEMBL5246346

O=C(NC1C2CCN(CC2)C1I)c1cc(Br)cc2oc(-c3ccccc3)nc12

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 6/20 0.44
CHRNB2 P17787 7/20 0.38
CHRNA7 P36544 7/20 0.38
CHRNA4 P43681 7/20 0.38
KCNH2 Q12809 3/20 0.38
HDAC6 Q9UBN7 1/20 0.36
USP30 Q70CQ3 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HIF1A Q16665 1/20 0.36
TOP2A P11388 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5248214 0.91 HTR3A (0.44) HTR3ACHRNB2CHRNA7CHRNA4KCNH2
SCHEMBL5245304 0.90 HTR3A (0.43) HTR3ACHRNB2CHRNA7CHRNA4KCNH2
SCHEMBL5246447 0.90 HTR3A (0.43) HTR3ACHRNB2CHRNA7CHRNA4KCNH2
SCHEMBL5247114 0.89 HTR3A (0.47) HTR3ACHRNB2CHRNA7CHRNA4KCNH2
SCHEMBL5244272 0.88 HTR3A (0.44) HTR3ACHRNB2CHRNA7CHRNA4KCNH2
SCHEMBL5243336 0.83 HTR3A (0.40) HTR3ACHRNB2CHRNA7CHRNA4KCNH2
SCHEMBL2957525 0.81 HTR3A (0.56) HTR3ACHRNA7KCNH2
SCHEMBL5245119 0.81 HTR3A (0.49) HTR3ACHRNB2CHRNA4KCNH2TOP2A
SCHEMBL5243252 0.81 HTR3A (0.46) HTR3ACHRNB2CHRNA7CHRNA4KCNH2
SCHEMBL5245030 0.80 HTR3A (0.59) HTR3ACHRNB2CHRNA7CHRNA4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1853597-A1 BENZOXAZOLE CARBOXAMIDES FOR TREATING CINV AND IBS-D AMR Technology, Inc. (US) 2007-11-14 EP disclosed
WO-2006089100-A1 BENZOXAZOLE CARBOXAMIDES FOR TREATING CINV AND IBS-D AMR TECHNOLOGY, INC. (US) 2006-08-24 WO disclosed