SCHEMBL5247498

SCHEMBL5247498

C=CCCCOc1cc(C(=O)NCC)ccc1-n1cc(C(=O)NCCCCO)nn1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMPD1 P17405 1/20 0.39
ACKR3 P25106 2/20 0.38
BRD4 O60885 1/20 0.37
POLB P06746 1/20 0.37
TP53 P04637 1/20 0.36
DRD2 P14416 4/20 0.35
DRD4 P21917 4/20 0.35
DRD3 P35462 4/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
PLK1 P53350 1/20 0.35
PLK3 Q9H4B4 1/20 0.35
PLK2 Q9NYY3 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5243944 0.97 SMPD1 (0.39) SMPD1ACKR3BRD4TP53MEN1
SCHEMBL5247607 0.92 KMT2A (0.43) ACKR3TP53NPC1RAB9AMEN1
SCHEMBL5250802 0.92 SMPD1 (0.38) SMPD1ACKR3BRD4TP53MEN1
SCHEMBL5244405 0.92 KMT2A (0.38) SMPD1ACKR3BRD4TP53NPC1
SCHEMBL5244829 0.92 BRD4 (0.37) SMPD1ACKR3BRD4TP53MEN1
SCHEMBL5247507 0.90 SMPD1 (0.38) SMPD1ACKR3BRD4TP53KMT2A
SCHEMBL5248452 0.90 BRD4 (0.36) SMPD1ACKR3BRD4TP53
SCHEMBL5248477 0.90 BRD4 (0.47) BRD4POLBTP53NPC1RAB9A
SCHEMBL5244268 0.89 PDK2 (0.35) SMPD1ACKR3POLBDRD2DRD4
SCHEMBL5248542 0.89 BRD4 (0.36) SMPD1ACKR3BRD4POLBTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1867331-A1 TRIAZOLE DERIVATIVE AND THE USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-12-19 EP disclosed