SCHEMBL5247607

SCHEMBL5247607

C=CCCCOc1cc(C(=O)NCC)ccc1-n1cc(C(=O)NCCCOCC)nn1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.43
MEN1 O00255 3/20 0.43
HPGD P15428 4/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
ALDH1A1 P00352 3/20 0.42
LMNA P02545 1/20 0.42
RAB9A P51151 2/20 0.41
NPC1 O15118 2/20 0.41
HTT P42858 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.39
MAPT P10636 4/20 0.39
PLA2G1B P04054 1/20 0.39
PAX8 Q06710 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
ATG4B Q9Y4P1 1/20 0.39
KDM4E B2RXH2 1/20 0.38
NAMPT P43490 1/20 0.38
ACKR3 P25106 1/20 0.37
TP53 P04637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5244405 0.96 KMT2A (0.38) KMT2AMEN1HPGDSMN1; SMN2ALDH1A1
SCHEMBL5243944 0.93 SMPD1 (0.39) KMT2AMEN1ACKR3TP53
SCHEMBL5247498 0.92 SMPD1 (0.39) KMT2AMEN1RAB9ANPC1ACKR3
SCHEMBL5244643 0.91 KMT2A (0.41) KMT2AMEN1HPGDSMN1; SMN2ALDH1A1
SCHEMBL5250802 0.91 SMPD1 (0.38) KMT2AMEN1ACKR3TP53
SCHEMBL5244829 0.91 BRD4 (0.37) KMT2AMEN1ACKR3TP53
SCHEMBL5245878 0.90 BRD4 (0.42) KMT2AHPGDSMN1; SMN2ALDH1A1RAB9A
SCHEMBL5248452 0.89 BRD4 (0.36) SMN1; SMN2MAPTACKR3TP53
SCHEMBL5247507 0.89 SMPD1 (0.38) KMT2ANAMPTACKR3TP53
SCHEMBL5248477 0.89 BRD4 (0.47) KMT2AMEN1HPGDSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1867331-A1 TRIAZOLE DERIVATIVE AND THE USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-12-19 EP disclosed