SCHEMBL5250802

SCHEMBL5250802

C=CCCCOc1cc(C(=O)NCC)ccc1-n1cc(C(=O)NCCOCCO)nn1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SMPD1 P17405 1/20 0.38
TP53 P04637 1/20 0.37
BRD4 O60885 5/20 0.36
ACKR3 P25106 2/20 0.35
PLK1 P53350 3/20 0.34
PLK3 Q9H4B4 3/20 0.34
PLK2 Q9NYY3 3/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
CNR2 P34972 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5244405 0.95 KMT2A (0.38) SMPD1TP53BRD4ACKR3MEN1
SCHEMBL5243944 0.93 SMPD1 (0.39) SMPD1TP53BRD4ACKR3PLK1
SCHEMBL5247498 0.92 SMPD1 (0.39) SMPD1TP53BRD4ACKR3PLK1
SCHEMBL5247607 0.91 KMT2A (0.43) TP53ACKR3MEN1KMT2A
SCHEMBL5244829 0.90 BRD4 (0.37) SMPD1TP53BRD4ACKR3MEN1
SCHEMBL5250028 0.90 SMPD1 (0.33) SMPD1TP53ACKR3
SCHEMBL5245878 0.89 BRD4 (0.42) TP53BRD4KMT2A
SCHEMBL5247507 0.89 SMPD1 (0.38) SMPD1TP53BRD4ACKR3KMT2A
SCHEMBL5248452 0.89 BRD4 (0.36) SMPD1TP53BRD4ACKR3CNR2
SCHEMBL5248542 0.88 BRD4 (0.36) SMPD1TP53BRD4ACKR3CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1867331-A1 TRIAZOLE DERIVATIVE AND THE USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-12-19 EP disclosed