SCHEMBL5248641

SCHEMBL5248641

NC(=O)Oc1cccn2cc(-c3cccc(C(F)(F)F)c3)nc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
MAPT P10636 2/20 0.43
NFKB1 P19838 2/20 0.43
NFKB2 Q00653 2/20 0.43
RELA Q04206 2/20 0.43
PKM P14618 1/20 0.43
EPHB4 P54760 7/20 0.43
CREBBP Q92793 1/20 0.42
F2RL3 Q96RI0 1/20 0.42
KMO O15229 2/20 0.41
ALDH1A3 P47895 1/20 0.41
DHODH Q02127 1/20 0.41
ABL1 P00519 1/20 0.41
EGFR P00533 1/20 0.41
PRKCB P05771 1/20 0.41
INSR P06213 1/20 0.41
LCK P06239 1/20 0.41
FYN P06241 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5249732 0.88 DHODH (0.46) NPC1RAB9ASMN1; SMN2MAPTNFKB1
SCHEMBL5250502 0.85 ALDH1A3 (0.48) NPC1RAB9ASMN1; SMN2MAPTNFKB1
SCHEMBL5251661 0.84 ALDH1A1 (0.49) NPC1RAB9ASMN1; SMN2MAPTNFKB1
SCHEMBL5251228 0.84 DHODH (0.53) NPC1RAB9ASMN1; SMN2MAPTNFKB1
SCHEMBL5252915 0.83 ALDH1A3 (0.46) NPC1RAB9ASMN1; SMN2MAPTNFKB1
SCHEMBL1419740 0.83 DHODH (0.52) NPC1RAB9ASMN1; SMN2MAPTNFKB1
SCHEMBL5251083 0.83 NPC1 (0.47) NPC1RAB9ASMN1; SMN2MAPTNFKB1
SCHEMBL5252624 0.82 DHODH (0.59) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL5251711 0.81 ALDH1A3 (0.60) NPC1RAB9ASMN1; SMN2MAPTNFKB1
SCHEMBL1419736 0.81 DHODH (0.64) NPC1RAB9ASMN1; SMN2MAPTNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1257551-B1 HETEROCYCLIC COMPOUNDS AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2007-09-05 EP disclosed