SCHEMBL5249909

SCHEMBL5249909

Fc1ccc(-c2scc(C3=CCN4CCC[C@H]4C3)c2-c2ccncc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 10/20 0.43
MAPK11 Q15759 5/20 0.43
MAPK13 O15264 2/20 0.35
MAPK12 P53778 2/20 0.35
CSNK1E P49674 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5249915 1.00 MAPK14 (0.43) MAPK14MAPK11MAPK13MAPK12CSNK1E
SCHEMBL5850103 0.82 MAPK14 (0.64) MAPK14MAPK11MAPK13MAPK12
SCHEMBL5849928 0.79 MAPK14 (0.61) MAPK14MAPK11MAPK13MAPK12
SCHEMBL5257670 0.78 MAPK14 (0.68) MAPK14MAPK11
SCHEMBL5257673 0.78 MAPK14 (0.68) MAPK14MAPK11
SCHEMBL5249451 0.77 MAPK14 (0.48) MAPK14MAPK11MAPK13MAPK12
SCHEMBL5247714 0.77 MAPK14 (0.48) MAPK14MAPK11MAPK13MAPK12
SCHEMBL5850032 0.73 MAPK11 (0.52) MAPK14MAPK11MAPK13MAPK12
SCHEMBL5851727 0.73 MAPK11 (0.51) MAPK14MAPK11MAPK13MAPK12
SCHEMBL5850082 0.71 MAPK11 (0.51) MAPK14MAPK11MAPK13MAPK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1361225-B1 COMPOUNDS SUBSTITUTED WITH BICYCLIC AMINO GROUPS SANKYO CO (JP) 2007-11-07 EP disclosed
US-7091352-B2 Compounds substituted with bicyclic amino groups SANKYO COMPANY, LIMITED (JP) 2006-08-15 US disclosed
US-20040147525-A1 Compounds substituted with bicyclic amino groups SANKYO COMPANY, LIMITED (JP) 2004-07-29 US disclosed
EP-1361225-A1 COMPOUNDS SUBSTITUTED WITH BICYCLIC AMINO GROUPS Sankyo Company, Limited (JP) 2003-11-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040147525-A1 Compounds substituted with bicyclic amino groups IL2, IL1B, IL4I1 MAPK14 1355/4885MAPK11 1447/4885MAPK13 2034/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.