SCHEMBL525148

SCHEMBL525148

O=S(=O)(O)C1CCCNC1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APLNR P35414 2/20 0.63
LMNA P02545 2/20 0.54
TSHR P16473 2/20 0.54
CYP3A4 P08684 1/20 0.54
GABRA1 P14867 1/20 0.54
GABRG2 P18507 1/20 0.54
NFKB1 P19838 1/20 0.54
GABRB3 P28472 1/20 0.54
GABRA5 P31644 1/20 0.54
GABRA3 P34903 1/20 0.54
GABRA2 P47869 1/20 0.54
GABRA6 Q16445 1/20 0.54
SLC6A1 P30531 2/20 0.43
SLC6A11 P48066 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
SLC6A13 Q9NSD5 1/20 0.43
KDM4E B2RXH2 1/20 0.42
MAPT P10636 1/20 0.42
KMT2A Q03164 1/20 0.42
ATM Q13315 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19815803 1.00 APLNR (0.63) APLNRLMNATSHRCYP3A4GABRA1
Hydrochloric Acid SCHEMBL28303066 0.98 APLNR (0.61) APLNRLMNATSHRCYP3A4GABRA1
SCHEMBL25873254 0.91 APLNR (0.53) APLNRLMNATSHRCYP3A4GABRA1
SCHEMBL3101278 0.86
SCHEMBL1546863 0.77 APLNR (1.00) APLNRLMNATSHRCYP3A4GABRA1
SCHEMBL18254434 0.77 APLNR (1.00) APLNRLMNATSHRCYP3A4GABRA1
SCHEMBL18254435 0.77 APLNR (1.00) APLNRLMNATSHRCYP3A4GABRA1
SCHEMBL19975528 0.77 APLNR (0.63) APLNRLMNATSHRCYP3A4GABRA1
SCHEMBL19565582 0.77 APLNR (0.63) APLNRLMNATSHRCYP3A4GABRA1
SCHEMBL6398719 0.77 APLNR (0.63) APLNRLMNATSHRCYP3A4GABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160193166-A1 ANTICONVULSIVE PHARMACEUTICAL COMPOSITIONS INSERM (INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE) (FR) 2016-07-07 US claimed
US-20100184707-A1 ANTICONVULSIVE PHARMACEUTICAL COMPOSITIONS INSERM (INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE) (FR) 2010-07-22 US claimed
US-11998602-B2 Methods for promoting myelination and for treating demyelinating diseases THE SCRIPPS RESEARCH INSTITUTE (US) 2024-06-04 US disclosed
US-11873291-B2 Quinoline cGAS antagonist compounds IMMUNESENSOR THERAPEUTICS, INC. (US) 2024-01-16 US disclosed
US-11873291-B2 Quinoline cGAS antagonist compounds IMMUNESENSOR THERAPEUTICS, INC. (US) 2024-01-16 US disclosed
US-20230246229-A1 ORGANIC SULFONATE ELECTROLYTE ADDITIVES FOR ZINC BATTERIES Octet Scientific, Inc. 2023-08-03 US disclosed
WO-2023141301-A1 ORGANIC SULFONATE ELECTROLYTE ADDITIVES FOR ZINC BATTERIES Octet Scientific, Inc. (US) 2023-07-27 WO disclosed
WO-2021107122-A1 HYPOXIA RESPONSE CONTROL BY SPECIFIC AMINO ACID OR AMINO ACID-LIKE SUBSTANCE 学校法人慶應義塾 2021-06-03 WO disclosed
US-20210023218-A1 METHODS FOR PROMOTING MYELINATION AND FOR TREATING DEMYELINATING DISEASES THE SCRIPPS RESEARCH INSTITUTE 2021-01-28 US disclosed
WO-2019172969-A1 METHODS FOR PROMOTING MYELINATION AND FOR TREATING DEMYELINATING DISEASES THE SCRIPPS RESEARCH INSTITUTE (US) 2019-09-12 WO disclosed
US-20190112656-A1 MITOCHONDRIAL BIOMARKER REFLECTING AGING KAWASAKI GAKUEN EDUCATIONAL FOUNDATION (JP) 2019-04-18 US disclosed
US-20160206579-A1 TAURINE OR TAURINE-LIKE SUBSTANCES FOR THE PREVENTION AND TREATMENT OF A DISEASE ASSOCIATED WITH RETINAL GANGLION CELL DEGENERATION INSERM (Institut National de la Santé et de la Recherche Médicale) (FR) 2016-07-21 US disclosed
US-20160193166-A1 ANTICONVULSIVE PHARMACEUTICAL COMPOSITIONS INSERM (INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE) (FR) 2016-07-07 US disclosed
US-20120027723-A1 TAURINE OR TAURINE-LIKE SUBSTANCES FOR THE PREVENTION AND TREATMENT OF A DISEASE ASSOCIATED WITH RETINAL GANGLION CELL DEGENERATION INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2012-02-02 US disclosed
EP-2393490-A1 TAURINE OR TAURINE-LIKE SUBSTANCES FOR THE PREVENTION AND TREATMENT OF A DISEASE ASSOCIATED WITH RETINAL GANGLION CELL DEGENERATION INSERM - Institut National de la Santé et de la Recherche Médicale (FR) 2011-12-14 EP disclosed
WO-2010089355-A1 TAURINE OR TAURINE-LIKE SUBSTANCES FOR THE PREVENTION AND TREATMENT OF A DISEASE ASSOCIATED WITH RETINAL GANGLION CELL DEGENERATION INSERM (Institut National de la Santé et de la Recherche Médicale) (FR) 2010-08-12 WO disclosed
EP-0666843-A1 SULFONYLALKANOYLAMINO HYDROXYETHYLAMINO SULFAMIC ACIDS USEFUL AS RETROVIRAL PROTEASE INHIBITORS G.D. SEARLE & CO. (US) 1995-08-16 EP disclosed
EP-0428831-B1 Process of preparation of pyridine-3-sulfonic acids RUETGERSWERKE AG (DE) 1994-06-08 EP disclosed
US-5082944-A Production of pyridine-3-sulfonic acid RUTGERSWERKE AG (DE) 1992-01-21 US disclosed
EP-0428831-A1 Process of preparation of pyridine-3-sulfonic acids RÜTGERSWERKE AKTIENGESELLSCHAFT (DE) 1991-05-29 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11873291-B2 Quinoline cGAS antagonist compounds CGAS, GLS2, GLS APLNR 3372/4885LMNA 1681/4885TSHR 2355/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.