SCHEMBL525272

SCHEMBL525272

C=COC(=O)N(O)CC

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4905114 0.79 MEN1 (0.43)
SCHEMBL17468762 0.77
SCHEMBL8213811 0.70
SCHEMBL7007254 0.70
SCHEMBL328721 0.70 CHRNB2 (0.32)
SCHEMBL1290917 0.69
SCHEMBL8928290 0.69
SCHEMBL27803238 0.68 TSHR (0.31)
SCHEMBL27660417 0.67 MEN1 (0.32)
SCHEMBL27263131 0.67 OPRK1 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 51 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103502317-B Macroinitiators containing hydrophobic segments 庄臣及庄臣视力保护公司 2017-02-08 CN claimed
WO-2024127114-A1 TRANSITION METAL COMPLEXES AS VISIBLE LIGHT ABSORBERS JOHNSON & JOHNSON VISION CARE, INC. (US) 2024-06-20 WO disclosed
WO-2023242688-A1 OPHTHALMIC DEVICES CONTAINING PHOTOSTABLE MIMICS OF MACULAR PIGMENT AND OTHER VISIBLE LIGHT FILTERS JOHNSON & JOHNSON VISION CARE, INC. (US) 2023-12-21 WO disclosed
EP-4263718-A1 PHOTOSTABLE MIMICS OF MACULAR PIGMENT Johnson & Johnson Vision Care, Inc. (US) 2023-10-25 EP disclosed
WO-2023119021-A1 CONTACT LENSES CONTAINING LIGHT ABSORBING REGIONS AND METHODS FOR THEIR PREPARATION JOHNSON & JOHNSON VISION CARE, INC. (US) 2023-06-29 WO disclosed
EP-4165015-A1 AMINO ACID-BASED POLYMERIZABLE COMPOUNDS AND OPHTHALMIC DEVICES PREPARED THEREFROM Johnson and Johnson Vision Care, Inc. (US) 2023-04-19 EP disclosed
EP-4165446-A1 IMIDAZOLIUM ZWITTERION POLYMERIZABLE COMPOUNDS AND OPHTHALMIC DEVICES INCORPORATING THEM Johnson & Johnson Vision Care, Inc. (US) 2023-04-19 EP disclosed
WO-2023052889-A1 AMIDE-FUNCTIONALIZED POLYMERIZATION INITIATORS AND THEIR USE IN THE MANUFACTURE OF OPHTHALMIC LENSES JOHNSON & JOHNSON VISION CARE, INC. (US) 2023-04-06 WO disclosed
EP-4121002-A1 OPHTHALMIC DEVICES CONTAINING TRANSITION METAL COMPLEXES AS HIGH ENERGY VISIBLE LIGHT FILTERS Johnson & Johnson Vision Care, Inc. (US) 2023-01-25 EP disclosed
EP-4022368-A1 CONTACT LENS DISPLAYING IMPROVED VISION ATTRIBUTES Johnson & Johnson Vision Care, Inc. (US) 2022-07-06 EP disclosed
EP-2598320-A1 OPHTHALMIC DEVICE MOLDS FORMED FROM WATER-SOLUBLE VINYL ALCOHOL COPOLYMER, OPHTHALMIC DEVICES MOLDED THEREIN, AND RELATED METHODS CooperVision International Holding Company, LP (BB) 2013-06-05 EP disclosed
EP-2598319-A1 OPHTHALMIC DEVICE MOLDS FORMED FROM HIGHLY AMORPHOUS VINYL ALCOHOL POLYMER, OPHTHALMIC DEVICES MOLDED THEREIN, AND RELATED METHODS CooperVision International Holding Company, LP (BB) 2013-06-05 EP disclosed
WO-2013033554-A1 BIOCOMPATIBLE MATERIAL VERTELLUS SPECIALTIES INC. (US) 2013-03-07 WO disclosed
WO-2013033553-A1 METHODS FOR PRODUCING BIOCOMPATIBLE MATERIALS VERTELLUS SPECIALTIES INC. (US) 2013-03-07 WO disclosed
WO-2012013948-A1 OPHTHALMIC DEVICE MOLDS FORMED FROM WATER-SOLUBLE VINYL ALCOHOL COPOLYMER, OPHTHALMIC DEVICES MOLDED THEREIN, AND RELATED METHODS GOODENOUGH NEIL (GB) 2012-02-02 WO disclosed
WO-2012013944-A1 OPHTHALMIC DEVICE MOLDS FORMED FROM HIGHLY AMORPHOUS VINYL ALCOHOL POLYMER, OPHTHALMIC DEVICES MOLDED THEREIN, AND RELATED METHODS GOODENOUGH NEIL (GB) 2012-02-02 WO disclosed
EP-1268410-A1 BETA-HYDROXY BUTENYL CARBAMATE, FUNCTIONAL OLIGOMERS AND COATINGS THEREFROM EASTMAN CHEMICAL COMPANY (US) 2003-01-02 EP disclosed
US-6465679-B2 (VINYL)-2-HYDROXYETHYL CARBAMATE; OLIGOMERS WITH A POLYISOCYANATE; CURABLE COATING COMPOSITIONS WITH MELAMINE-FORMALDEHYDE RESIN; LOW SOLUTION VISCOSITY, FOR USE IN HIGH SOLIDS COATINGS EASTMAN CHEMICAL COMPANY 2002-10-15 US disclosed
US-20020040110-A1 Carbamate functional oligomers and coatings therefrom EASTMAN CHEMICAL COMPANY 2002-04-04 US disclosed
WO-2001049658-A1 BETA-HYDROXY BUTENYL CARBAMATE, FUNCTIONAL OLIGOMERS AND COATINGS THEREFROM EASTMAN CHEMICAL COMPANY (US) 2001-07-12 WO disclosed