SCHEMBL5253618

SCHEMBL5253618

CN1CCN(Cc2cccc(Br)n2)CC1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.54
CXCR4 P61073 2/20 0.49
HRH4 Q9H3N8 2/20 0.48
MC4R P32245 1/20 0.47
KDM4E B2RXH2 2/20 0.45
TDP1 Q9NUW8 1/20 0.45
ACHE P22303 1/20 0.45
CHKA P35790 2/20 0.43
DRD2 P14416 1/20 0.43
DRD3 P35462 1/20 0.43
LMNA P02545 1/20 0.41
CA2 P00918 1/20 0.41
NCF1 P14598 1/20 0.41
PRMT6 Q96LA8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22205248 0.88 CXCR4 (0.61) CXCR4HRH4MC4RKDM4ECHKA
SCHEMBL29462386 0.87 FAAH (0.54) FAAHCXCR4KDM4ETDP1ACHE
SCHEMBL5255062 0.87 FAAH (0.54) FAAHCXCR4KDM4ETDP1ACHE
Hydrochloric Acid SCHEMBL29604571 0.86 CXCR4 (0.59) CXCR4HRH4MC4RKDM4ECHKA
Bromide SCHEMBL29604007 0.86 CXCR4 (0.59) CXCR4HRH4MC4RKDM4ECHKA
SCHEMBL839038 0.83 FAAH (0.53) FAAHCXCR4HRH4KDM4ETDP1
SCHEMBL13940602 0.83 FAAH (0.51) FAAHCXCR4KDM4ETDP1ACHE
SCHEMBL14851189 0.81 HTR3E (0.53) CXCR4HRH4MC4RKDM4EACHE
SCHEMBL15980623 0.81 CXCR4 (0.46) FAAHCXCR4HRH4MC4RKDM4E
SCHEMBL840048 0.81 KMT2A (0.59) FAAHCXCR4KDM4EACHEDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268431-B1 3-CYANOQUINOLINES,3-CYANO-1,6-NAPHTHYRIDINES, AND 3-CYANO-1,7-NAPHTHYRIDINES AS PROTEIN KINASE INHIBITORS WYETH CORP (US) 2007-08-29 EP disclosed