SCHEMBL5255165

SCHEMBL5255165

CCN(CC)CCCOc1ccc2c(c1)c(C1=C(c3cccc4ccoc34)C(=O)NC1=O)cn2C(C)C

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.45
GSK3B P49841 6/20 0.40
GSK3A P49840 4/20 0.40
ACHE P22303 3/20 0.38
XDH P47989 1/20 0.36
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
LYN P07948 1/20 0.35
SRC P12931 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5252434 0.98 SIGMAR1 (0.45) SIGMAR1GSK3BGSK3AACHEMAOA
SCHEMBL5252064 0.90 GSK3B (0.41) GSK3BGSK3A
SCHEMBL5257697 0.90 GSK3B (0.40) GSK3BGSK3AMAOAMAOB
Hydrochloric Acid SCHEMBL5256878 0.89 SIGMAR1 (0.44) SIGMAR1GSK3BGSK3AACHEXDH
SCHEMBL5256883 0.89 GSK3B (0.42) GSK3BGSK3A
Hydrochloric Acid SCHEMBL5254194 0.89 SIGMAR1 (0.43) SIGMAR1GSK3BGSK3AACHELYN
SCHEMBL5253874 0.88 GSK3B (0.41) GSK3BGSK3A
SCHEMBL5252491 0.88 SIGMAR1 (0.45) SIGMAR1GSK3BGSK3AACHEMAOA
Hydrochloric Acid SCHEMBL5255252 0.85 SIGMAR1 (0.42) SIGMAR1GSK3BGSK3AMAOAMAOB
Hydrochloric Acid SCHEMBL5253479 0.85 GSK3B (0.47) SIGMAR1GSK3BGSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487822-B1 PYRROLE-2,5-DIONE DERIVATIVES AND THEIR USE AS GSK-3 INHIBITORS LILLY CO ELI (US) 2007-08-01 EP disclosed
CN-1639152-A Pyrrole-2, 5-dione derivatives and their use as GSK-3 inhibitors LILLY CO ELI (US) 2005-07-13 CN disclosed