SCHEMBL5255808

SCHEMBL5255808

Fc1ccc2[nH]nc(Nc3nc(-c4ccccc4)nc4c3CCCC4)c2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 1/20 0.52
EGFR P00533 3/20 0.49
PDE4B Q07343 2/20 0.47
FADS1 O60427 2/20 0.44
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
HTR2B P41595 1/20 0.43
GSK3A P49840 2/20 0.42
GSK3B P49841 2/20 0.42
AURKA O14965 1/20 0.42
AURKB Q96GD4 1/20 0.42
LMNA P02545 2/20 0.41
MEN1 O00255 1/20 0.41
MAPT P10636 1/20 0.41
KMT2A Q03164 1/20 0.41
BCHE P06276 3/20 0.40
ACHE P22303 3/20 0.40
GRIN1 Q05586 3/20 0.40
GRIN2A Q12879 3/20 0.40
VCP P55072 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL786842 0.88 HTR2A (0.57) IGF1REGFRFADS1HTR2AHTR2C
SCHEMBL786092 0.87 IGF1R (0.49) IGF1REGFRPDE4BFADS1VCP
SCHEMBL786744 0.85 FADS1 (0.45) IGF1REGFRFADS1GSK3AGSK3B
SCHEMBL13107334 0.85 EGFR (0.42) IGF1REGFRPDE4BFADS1GSK3A
SCHEMBL786140 0.84 IGF1R (0.51) IGF1REGFRPDE4BHTR2AHTR2C
SCHEMBL14164030 0.84 EGFR (0.42) IGF1REGFRPDE4BFADS1GSK3A
SCHEMBL785653 0.84 USP1 (0.46) IGF1REGFRFADS1GSK3AGSK3B
SCHEMBL786233 0.84 FADS1 (0.46) IGF1REGFRFADS1GSK3AGSK3B
SCHEMBL785480 0.84 USP1 (0.45) IGF1REGFRFADS1GSK3AGSK3B
SCHEMBL802419 0.84 EGFR (0.43) IGF1REGFRFADS1GSK3AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1318814-B1 TRIAZOLE COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS VERTEX PHARMA (US) 2007-05-30 EP disclosed