SCHEMBL5255876

SCHEMBL5255876

C=CCOc1cccc2c1C(NOCc1ccccc1)CNC2C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
LIG1 P18858 1/20 0.37
HTR1A P08908 2/20 0.34
SLC6A2 P23975 2/20 0.34
SLC6A4 P31645 2/20 0.34
SLC6A3 Q01959 2/20 0.34
NPC1 O15118 2/20 0.33
POLB P06746 1/20 0.33
RAB9A P51151 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CXCR5 P32302 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
BCHE P06276 2/20 0.32
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5253702 0.92 HTR1A (0.38) MEN1KMT2AHTR1ASLC6A2SLC6A4
SCHEMBL4139603 0.90 MEN1 (0.39) MEN1KMT2ALIG1NPC1POLB
SCHEMBL4136367 0.83 BCHE (0.42) NPC1RAB9AALDH1A1BCHEGAA
SCHEMBL5256420 0.83 BCHE (0.42) NPC1RAB9AALDH1A1BCHEGAA
SCHEMBL5185631 0.82 KMT2A (0.39) MEN1KMT2AHTR1ASLC6A2SLC6A4
SCHEMBL4696919 0.81 MEN1 (0.36) MEN1KMT2ALIG1HTR1ASLC6A2
SCHEMBL5330841 0.80 TSHR (0.40) HTR1ASLC6A2SLC6A4SLC6A3NPC1
SCHEMBL5257111 0.78 TSHR (0.38) MEN1KMT2ALIG1POLBALDH1A1
SCHEMBL5186922 0.75 BCHE (0.38) NPC1POLBRAB9AALDH1A1BCHE
SCHEMBL4144345 0.75 MEN1 (0.38) MEN1KMT2ALIG1POLBCXCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1798231-A2 Intermediate products for the preparation of antibacterial compounds NOVEXEL (FR) 2007-06-20 EP disclosed
EP-1399444-B1 NOVEL HETEROCYCLIC COMPOUNDS, METHOD FOR PREPARING SAME AND USE THEREOF AS MEDICINES, IN PARTICULAR AS ANTI-BACTERIAL AGENTS NOVEXEL (FR) 2007-04-11 EP disclosed
EP-1399444-A2 NOVEL HETEROCYCLIC COMPOUNDS, METHOD FOR PREPARING SAME AND USE THEREOF AS MEDICINES, IN PARTICULAR AS ANTI-BACTERIAL AGENTS Aventis Pharma S.A. (FR) 2004-03-24 EP disclosed
WO-2002100860-A2 HETEROCYCLIC COMPOUNDS, METHOD FOR PREPARING SAME AND USE THEREOF AS MEDICINES, IN PARTICULAR AS ANTI-BACTERIAL AGENTS AVENTIS PHARMA S.A. (FR) 2002-12-19 WO disclosed