SCHEMBL4696919

SCHEMBL4696919

C=CCOc1cccc2c1C(NOCc1ccccc1)CN(C(=O)O)C2C(=O)O

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
LIG1 P18858 1/20 0.35
FAAH O00519 3/20 0.35
GYS1 P13807 1/20 0.33
ACE P12821 5/20 0.33
MGLL Q99685 1/20 0.33
NPC1 O15118 2/20 0.32
POLB P06746 1/20 0.32
RAB9A P51151 1/20 0.32
HTR1A P08908 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
PTGER1 P34995 1/20 0.32
PTGER4 P35408 1/20 0.32
PTGER3 P43115 1/20 0.32
PTGER2 P43116 1/20 0.32
SIRT1 Q96EB6 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4144345 0.90 MEN1 (0.38) MEN1KMT2ALIG1FAAHACE
SCHEMBL4142735 0.83 NPC1 (0.40) GYS1NPC1POLBRAB9A
SCHEMBL5255838 0.83 NPC1 (0.40) GYS1NPC1POLBRAB9A
SCHEMBL5255462 0.83 HTR1A (0.36) NPC1HTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL5255876 0.81 MEN1 (0.37) MEN1KMT2ALIG1NPC1POLB
SCHEMBL5254943 0.79 NPC1 (0.38) ACENPC1RAB9A
SCHEMBL5253676 0.77 ACE (0.36) LIG1FAAHACEPOLB
SCHEMBL4139603 0.75 MEN1 (0.39) MEN1KMT2ALIG1NPC1POLB
SCHEMBL5186348 0.75 POLB (0.38) FAAHNPC1POLBRAB9A
SCHEMBL5187180 0.74 KMT2A (0.38) MEN1KMT2AHTR1ASLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569935-B1 HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREOF AND USE OF SAME AS MEDICAMENTS, SUCH AS ANTI-BACTERIAL MEDICAMENTS AND BETA-LACTAMASE INHIBITORS NOVEXEL (FR) 2008-08-20 EP disclosed
EP-1798231-A2 Intermediate products for the preparation of antibacterial compounds NOVEXEL (FR) 2007-06-20 EP disclosed
EP-1399444-B1 NOVEL HETEROCYCLIC COMPOUNDS, METHOD FOR PREPARING SAME AND USE THEREOF AS MEDICINES, IN PARTICULAR AS ANTI-BACTERIAL AGENTS NOVEXEL (FR) 2007-04-11 EP disclosed