SCHEMBL5256405

SCHEMBL5256405

Cn1cncc1CNc1ccc(-c2nc3cc(Br)cnc3[nH]2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.34
RAB9A P51151 3/20 0.34
KMT2A Q03164 2/20 0.34
MAP3K8 P41279 1/20 0.34
HPSE Q9Y251 2/20 0.34
AURKA O14965 2/20 0.33
BRD4 O60885 1/20 0.33
KDR P35968 4/20 0.33
ABL1 P00519 2/20 0.33
RET P07949 2/20 0.33
CDK7 P50613 2/20 0.33
CDK5 Q00535 2/20 0.33
PRKAA1 Q13131 2/20 0.33
AURKB Q96GD4 2/20 0.33
CLK4 Q9HAZ1 2/20 0.33
IDH1 O75874 1/20 0.32
MEN1 O00255 1/20 0.32
GFER P55789 1/20 0.32
ITK Q08881 2/20 0.31
MET P08581 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL4840394 0.91 SYK (0.35) NPC1RAB9AKMT2AMAP3K8HPSE
SCHEMBL4834899 0.78 MMP2 (0.43) NPC1RAB9AKMT2AHPSESMN1; SMN2
SCHEMBL4837685 0.78 TAAR1 (0.47)
SCHEMBL5258759 0.78 NPC1 (0.38) NPC1RAB9AKMT2AHPSEAURKA
SCHEMBL5259468 0.78 NPC1 (0.34) NPC1RAB9AKMT2AHPSEAURKA
SCHEMBL5261764 0.77 HPSE (0.39) NPC1RAB9AKMT2AHPSETP53
SCHEMBL5261107 0.77 NPC1 (0.62) NPC1RAB9AKMT2AMEN1GFER
SCHEMBL5257452 0.76 NPC1 (0.34) NPC1RAB9AKMT2AHPSEAURKA
SCHEMBL5259906 0.76 LMNA (0.43) NPC1RAB9AKMT2AHPSEKDR
SCHEMBL4844738 0.76 HPSE (0.41) NPC1RAB9AHPSEABL1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539759-B1 NOVEL IMIDAZOPYRIDINES AND THEIR USE ASTRAZENECA AB (SE) 2007-08-15 EP claimed