SCHEMBL5258265

SCHEMBL5258265

CCCOC(=O)N1CCc2c(sc(N)c2C(=O)O)C1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 6/20 0.67
MAPT P10636 12/20 0.57
ALDH1A1 P00352 8/20 0.57
KDM4E B2RXH2 6/20 0.57
RAD52 P43351 1/20 0.57
GAA P10253 4/20 0.57
MEN1 O00255 7/20 0.51
KMT2A Q03164 7/20 0.51
HPGD P15428 6/20 0.48
ALOX15 P16050 3/20 0.47
HSD17B10 Q99714 2/20 0.47
LMNA P02545 2/20 0.46
GLA P06280 1/20 0.45
ADORA3 P0DMS8 1/20 0.45
PDE4D Q08499 1/20 0.45
NPSR1 Q6W5P4 5/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
TSHR P16473 2/20 0.44
PKM P14618 1/20 0.44
BLM P54132 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4134826 0.85 ADORA1 (0.74) ADORA1MAPTALDH1A1KDM4EGAA
SCHEMBL10855842 0.83 ADORA1 (0.59) ADORA1MAPTALDH1A1KDM4ERAD52
SCHEMBL970355 0.81 ADORA1 (0.83) ADORA1MAPTALDH1A1KDM4EGAA
SCHEMBL8288691 0.81 ADORA1 (0.68) ADORA1MAPTALDH1A1KDM4EGAA
SCHEMBL4131894 0.81 ALDH1A1 (0.50) ADORA1MAPTALDH1A1KDM4EMEN1
SCHEMBL3499018 0.81 ADORA1 (1.00) ADORA1MAPTALDH1A1KDM4ERAD52
SCHEMBL19475110 0.81 MAPT (0.72) ADORA1MAPTALDH1A1KDM4ERAD52
SCHEMBL16007549 0.80 ADORA1 (0.72) ADORA1MAPTALDH1A1KDM4EGAA
SCHEMBL10856568 0.79 ADORA1 (0.69) ADORA1MAPTALDH1A1KDM4ERAD52
SCHEMBL29229875 0.79 ADORA1 (0.68) ADORA1MAPTALDH1A1KDM4ERAD52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1802634-A2 THIOPHENS AND THEIR USE AS ANTI-TUMOR AGENTS Compass Pharmaceuticals LLC (US) 2007-07-04 EP claimed
WO-2006044826-A2 THIOPHENS AND THEIR USE AS ANTI-TUMOR AGENTS COMPASS PHARMACEUTICALS LLC (US) 2006-04-27 WO claimed
EP-1802634-A2 THIOPHENS AND THEIR USE AS ANTI-TUMOR AGENTS Compass Pharmaceuticals LLC (US) 2007-07-04 EP disclosed
WO-2006044826-A2 THIOPHENS AND THEIR USE AS ANTI-TUMOR AGENTS COMPASS PHARMACEUTICALS LLC (US) 2006-04-27 WO disclosed