SCHEMBL5258641

SCHEMBL5258641

CC(C)(C)OC(=O)NC(C)(I)c1ccc(Br)cc1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.49
RAB9A P51151 4/20 0.49
RECQL P46063 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
AAK1 Q2M2I8 8/20 0.41
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
GAA P10253 1/20 0.38
HTT P42858 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
FPR3 P25089 1/20 0.36
FPR2 P25090 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3797749 1.00 NPC1 (0.49) NPC1RAB9ARECQLSMN1; SMN2AAK1
SCHEMBL3670192 1.00 NPC1 (0.49) NPC1RAB9ARECQLSMN1; SMN2AAK1
SCHEMBL5505022 0.84 EPHX2 (0.37) NPC1RAB9ARECQLSMN1; SMN2AAK1
SCHEMBL1141998 0.83 NPC1 (0.51) NPC1RAB9ARECQLSMN1; SMN2AAK1
SCHEMBL3953935 0.80 DHODH (0.38) NPC1RAB9AAAK1CTSSCTSK
SCHEMBL3650222 0.80 RAB9A (0.43) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL1208679 0.79 NPC1 (0.48) NPC1RAB9ARECQLSMN1; SMN2AAK1
SCHEMBL5503662 0.79 ALDH1A1 (0.46) NPC1RAB9ARECQLSMN1; SMN2MEN1
SCHEMBL1141266 0.78 NPC1 (0.47) NPC1RAB9ARECQLSMN1; SMN2AAK1
SCHEMBL1433131 0.77 NPC1 (0.43) NPC1RAB9ARECQLSMN1; SMN2AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781662-A1 INHIBITORS OF HEPATITIS C VIRUS RNA-DEPENDENT RNA POLYMERASE, AND COMPOSITIONS AND TREATMENTS USING THE SAME Pfizer, Inc. (US) 2007-05-09 EP disclosed
WO-2006018725-A1 INHIBITORS OF HEPATITIS C VIRUS RNA-DEPENDENT RNA POLYMERASE, AND COMPOSITIONS AND TREATMENTS USING THE SAME PFIZER INC. (US) 2006-02-23 WO disclosed