SCHEMBL525883

SCHEMBL525883

C=CCc1ccc(O)c(-c2ccc(OC(CCNC)c3ccccc3)c(CC=C)c2)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 11/20 0.59
GABRB2 P47870 11/20 0.59
ALOX5 P09917 7/20 0.59
CNR2 P34972 4/20 0.59
CNR1 P21554 2/20 0.54
KMT2A Q03164 3/20 0.52
MEN1 O00255 2/20 0.52
POLB P06746 1/20 0.52
GAA P10253 1/20 0.52
MAPT P10636 1/20 0.52
GABRB1 P18505 1/20 0.52
RXRA P19793 1/20 0.52
GABRA5 P31644 1/20 0.52
GABRA3 P34903 1/20 0.52
GABRA2 P47869 1/20 0.52
ACE2 Q9BYF1 1/20 0.52
SIRT3 Q9NTG7 1/20 0.52
CYP1A2 P05177 4/20 0.43
CYP3A4 P08684 4/20 0.43
CYP2D6 P10635 4/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL526406 0.99 GABRA1 (0.58) GABRA1GABRB2ALOX5CNR2CNR1
SCHEMBL526354 0.93 GABRA1 (0.57) GABRA1GABRB2ALOX5CNR2CNR1
Hydrochloric Acid SCHEMBL726872 0.92 GABRA1 (0.56) GABRA1GABRB2ALOX5CNR2CNR1
SCHEMBL525534 0.88 GABRA1 (0.54) GABRA1GABRB2ALOX5CNR2CNR1
SCHEMBL525518 0.88 GABRA1 (0.56) GABRA1GABRB2ALOX5CNR2CNR1
Hydrochloric Acid SCHEMBL530274 0.88 GABRA1 (0.53) GABRA1GABRB2ALOX5CNR2CNR1
Hydrochloric Acid SCHEMBL530310 0.87 GABRA1 (0.55) GABRA1GABRB2ALOX5CNR2CNR1
SCHEMBL525888 0.86 GABRA1 (0.56) GABRA1GABRB2ALOX5CNR2CNR1
Hydrochloric Acid SCHEMBL725496 0.85 GABRA1 (0.55) GABRA1GABRB2ALOX5CNR2CNR1
SCHEMBL528431 0.84 GABRA1 (0.55) GABRA1GABRB2ALOX5CNR2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2423181-A1 Multitarget substituted biphenyl diol derivatives PROUS INSTITUTE FOR BIOMEDICAL RESEARCH S.A. (ES) 2012-02-29 EP claimed
WO-2012013691-A1 MULTITARGET SUBSTITUTED BIPHENYL DIOL DERIVATIVES PROUS INSTITUTE FOR BIOMEDICAL RESEARCH, S.A. (ES) 2012-02-02 WO claimed
EP-2423181-A1 Multitarget substituted biphenyl diol derivatives PROUS INSTITUTE FOR BIOMEDICAL RESEARCH S.A. (ES) 2012-02-29 EP disclosed
EP-2423181-A1 Multitarget substituted biphenyl diol derivatives PROUS INSTITUTE FOR BIOMEDICAL RESEARCH S.A. (ES) 2012-02-29 EP disclosed