SCHEMBL5259197

SCHEMBL5259197

Fc1ccccc1-c1nc(Nc2n[nH]c3ccc(C(F)(F)F)cc23)c2ccccc2n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 6/20 0.53
KMT2A Q03164 6/20 0.53
MAPT P10636 5/20 0.52
POLB P06746 2/20 0.52
MAPK1 P28482 1/20 0.52
LMNA P02545 3/20 0.50
TP53 P04637 2/20 0.50
ABCG2 Q9UNQ0 4/20 0.49
USP1 O94782 3/20 0.48
WDR48 Q8TAF3 3/20 0.48
FADS1 O60427 1/20 0.48
ALDH1A1 P00352 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
KDM4E B2RXH2 2/20 0.46
HTT P42858 1/20 0.46
GBA1 P04062 2/20 0.46
TRPA1 O75762 1/20 0.45
CHEK1 O14757 1/20 0.44
CHEK2 O96017 1/20 0.44
CYP1A2 P05177 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL786427 0.90 USP1 (0.61) MEN1KMT2AMAPTLMNATP53
SCHEMBL785470 0.89 FADS1 (0.53) MEN1KMT2AMAPTMAPK1LMNA
SCHEMBL786256 0.82 USP1 (0.64) MEN1KMT2AMAPTLMNATP53
SCHEMBL785772 0.82 USP1 (0.61) MEN1KMT2AMAPTLMNATP53
SCHEMBL1083832 0.80 USP1 (0.47) MEN1KMT2AMAPTPOLBMAPK1
SCHEMBL10268959 0.80 USP1 (0.47) MEN1KMT2AMAPTPOLBMAPK1
SCHEMBL801914 0.79 FADS1 (0.49) MEN1KMT2AMAPTPOLBMAPK1
SCHEMBL786042 0.79 CYP1A2 (0.58) MEN1KMT2AMAPTLMNATP53
SCHEMBL785641 0.79 USP1 (0.56) MEN1KMT2AMAPTLMNATP53
SCHEMBL786391 0.79 CYP1A2 (0.57) MEN1KMT2AMAPTLMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1318814-B1 TRIAZOLE COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS VERTEX PHARMA (US) 2007-05-30 EP disclosed