SCHEMBL5259392

SCHEMBL5259392

CCc1ccc2[nH]c(C(=O)N[C@H]3CCCC[C@H]3C(=O)O)cc2c1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.54
PYGL P06737 3/20 0.51
PYGM P11217 1/20 0.51
NPC1 O15118 2/20 0.49
MAPT P10636 1/20 0.49
MLLT1 Q03111 1/20 0.49
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
RAB9A P51151 1/20 0.47
EHMT2 Q96KQ7 1/20 0.44
CCKBR P32239 1/20 0.42
TSHR P16473 1/20 0.42
F10 P00742 6/20 0.42
F2 P00734 2/20 0.42
HPGD P15428 1/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
SMYD3 Q9H7B4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5258969 0.84 MLLT1 (0.53) MLLT1CCKBRF10F2SMYD3
SCHEMBL6834814 0.84 MLLT1 (0.53) MLLT1CCKBRF10F2SMYD3
SCHEMBL6832859 0.83 MLLT1 (0.52) PYGLPYGMMLLT1MEN1KMT2A
SCHEMBL7069488 0.83 SMYD3 (0.61) PYGLMLLT1EHMT2F10F2
SCHEMBL7067623 0.83 MLLT1 (0.72) KDM4EPYGLPYGMMLLT1MEN1
SCHEMBL5256226 0.82 KDM4E (0.43) KDM4EPYGLPYGMNPC1MAPT
SCHEMBL6833159 0.82 KDM4E (0.43) KDM4EPYGLPYGMNPC1MAPT
SCHEMBL5256019 0.81 CCKBR (0.57) KDM4EPYGLPYGMNPC1MAPT
SCHEMBL27558367 0.81 CCKBR (0.57) KDM4EPYGLPYGMNPC1MAPT
SCHEMBL16842009 0.80 MLLT1 (0.51) KDM4EPYGLPYGMMLLT1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1453801-B1 SUBSTITUTED 2-AMINO-CYCLOALKANECARBOXAMIDES AND THEIR USE AS CYSTEINE PROTEASE INHIBITORS HOFFMANN LA ROCHE (CH) 2007-03-21 EP disclosed