SCHEMBL5259676

SCHEMBL5259676

Cc1ccccc1C(O)C(=N)N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.43
ALDH1A1 P00352 2/20 0.40
GAA P10253 2/20 0.40
ACP3 P15309 1/20 0.38
TSHR P16473 1/20 0.36
ACHE P22303 1/20 0.36
CYP3A4 P08684 2/20 0.33
SLC6A2 P23975 2/20 0.33
SLC6A4 P31645 2/20 0.33
SLC6A3 Q01959 2/20 0.33
CYP1A2 P05177 1/20 0.33
F2 P00734 1/20 0.33
F10 P00742 1/20 0.33
F12 P00748 1/20 0.33
F7 P08709 1/20 0.33
F3 P13726 1/20 0.33
PKM P14618 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CYP2D6 P10635 1/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7449447 0.81 ESR1 (0.45) ESR1ALDH1A1GAAACP3TSHR
SCHEMBL1197054 0.79 ALDH1A1 (0.47) ESR1ALDH1A1GAAACP3TSHR
SCHEMBL9310523 0.79 ALDH1A1 (0.47) ESR1ALDH1A1GAAACP3TSHR
SCHEMBL11903290 0.79 ALDH1A1 (0.47) ESR1ALDH1A1GAAACP3TSHR
SCHEMBL13993318 0.77 ESR1 (0.59) ESR1ALDH1A1GAAACP3TSHR
SCHEMBL30507724 0.74 ESR1 (0.56) ESR1ALDH1A1GAAACP3TSHR
SCHEMBL1669099 0.73 ESR1 (0.50) ESR1ALDH1A1GAAACP3TSHR
SCHEMBL124623 0.72 ESR1 (0.45) ESR1ALDH1A1GAAACP3TSHR
SCHEMBL168464 0.72 LMNA (0.52) ESR1ALDH1A1GAAACP3TSHR
SCHEMBL21552683 0.72 ESR1 (0.45) ESR1ALDH1A1GAAACP3TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765795-A2 ALKYNYL DERIVATIVES AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS Addex Pharmaceuticals SA (CH) 2007-03-28 EP disclosed
WO-2005123703-A2 ALKYNYL DERIVATIVES AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS ADDEX PHARMACEUTICALS SA (CH) 2005-12-29 WO disclosed