SCHEMBL5260072

SCHEMBL5260072

O=C(N[C@H]1CCCC[C@H]1C(=O)O)c1cnc2ccccc2n1

nearest known ligand 0.70

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.53
ALDH1A1 P00352 1/20 0.50
HPGD P15428 1/20 0.50
ALOX15 P16050 1/20 0.50
HSD17B10 Q99714 1/20 0.50
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
HCRTR1 O43613 2/20 0.47
HCRTR2 O43614 2/20 0.47
PTK2 Q05397 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5256081 1.00 SMN1; SMN2 (0.53) SMN1; SMN2ALDH1A1HPGDALOX15HSD17B10
SCHEMBL28746033 1.00 SMN1; SMN2 (0.53) SMN1; SMN2ALDH1A1HPGDALOX15HSD17B10
SCHEMBL5256700 0.83 SSTR3 (0.58) SMN1; SMN2ALDH1A1HPGDNPC1RAB9A
SCHEMBL5255157 0.83 SSTR3 (0.58) SMN1; SMN2ALDH1A1HPGDNPC1RAB9A
SCHEMBL14565583 0.83 SSTR3 (0.58) SMN1; SMN2ALDH1A1HPGDNPC1RAB9A
SCHEMBL6205464 0.82 CNR1 (0.58) SMN1; SMN2ALDH1A1HPGDALOX15HSD17B10
SCHEMBL6083987 0.81 CNR1 (0.60) SMN1; SMN2ALDH1A1HPGDALOX15HSD17B10
SCHEMBL6084329 0.81 CNR1 (0.60) SMN1; SMN2ALDH1A1HPGDALOX15HSD17B10
SCHEMBL6832879 0.80 HPGDS (0.57)
SCHEMBL6083965 0.80 TAS1R3 (0.53) SMN1; SMN2ALDH1A1HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1453801-B1 SUBSTITUTED 2-AMINO-CYCLOALKANECARBOXAMIDES AND THEIR USE AS CYSTEINE PROTEASE INHIBITORS HOFFMANN LA ROCHE (CH) 2007-03-21 EP disclosed
US-6747053-B2 Heteroaryl nitriles ROCHE PALO ALTO LLC 2004-06-08 US disclosed